4 Benzyloxy 2 trifluoromethoxy phenylboronic acid 3 Bromo 4 methoxyphenylboronic acid pinacol ester 5 4 Morpholinylmethyl thiophene 2 boronic acid pinacol ester 3 Bromo 4 fluorophenylboronic acid pinacol ester 2 5 Difluoro 6 methylbenzeneboronic acid pinacol ester 3 Cyclobutylphenylboronic acid 3 Hydroxy 2 methylphenylboronic acid 2 Methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 Cyano 3 ethylphenylboronic acid 2 6 Dimethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 4 Cyclobutylphenyl boronic acid 3 Methoxy 4 phenoxyphenylboronic acid 2 Bromo 5 trifluoromethylphenylboronic acid pinacol ester 5 Butylthiophen 2 boronic acid 4 Fluorobenzofuran 7 boronic acid 5 Bromo 2 fluorophenylboronic acid pinacol ester 2 2 5 bis Trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 Bis trifluoromethyl phenylboronic acid pinacol ester 2 Bromothiazole 5 boronic acid pinacol ester 4 Cyano 2 fluorobenzeneboronic acid pinacol ester 2 2 Bromo 5 chlorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 Dichloro 4 trifluoromethyl phenylboronic acid 2 Methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 4 Bromo 3 5 dimethylphenylboronic acid pinacol ester 2 Chloro 4 phenoxy phenylboronic acid pinacol ester 4 Chloro 2 fluoro 5 methylbenzoic acid 2 Fluoro 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Fluoro 3 formylphenylboronic acid pinacol ester 2 Bromo 5 carboxyphenylboronic acid 3 Hydroxy 2 methoxypyridine 5 boronic acid pinacol ester

5 Hexylthiopheneboronic acid pinacol ester 5 Hydroxy 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 5 Fluoro 4 methylpyridin 3 yl boronic acid 3 Fluoro 5 pyrrolidino phenylboronic acid pinacol ester 3 Cyano 2 methylphenylboronic acid 3 Ffluoro N N dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 4 Methyl 3 phenylbenzenboronic acid 2 Dimethylamino 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl cyclohex 3 enol 2 Hydroxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzenemethanol 3 Amino 4 methylphenylboronic acid pinacol ester 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 3 trifluoromethyl aniline 2 6 difluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzenemethanol 4 Tert butylaminomethyl phenylboronic acid pinacol ester 4 Cyano 2 methylphenylboronic acid pinacol ester 5 Bromo 2 methylphenylboronic acid pinacol ester 4 Dimethylamino 5 formylphenylboronic acid pinacol ester 2 Fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 3 Methoxy 4 methoxymethoxy phenylboronic acid 3 Chloro 5 cyanophenylboronic acid pinacol ester 7 Methyl 1H indazole 4 boronic acid pinacol ester 3 Chloro 2 fluoropyridne 5 boronic acid pinacol ester 3 4 Boc 1 piperazinylmethyl benzeneboronic acid pinacol ester 2 Chloro 6 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 3 Chloro 4 N N dimethylamino phenylboronic acid pinacol ester 2 Hydroxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 2 2 Methoxyethoxy pyridine 5 boronic acid 2 Ethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 3 Bromo 5 chloro 2 6 difluorophenylboronic acid pinaco ester 4 Amino 3 trifluoromethoxy phenylboronic acid pinacol ester

4 Bromo 3 methoxyphenylboronic acid 2 Amino 5 isopropylphenylboronic acid pinacol ester 4 Trifluoromethoxy 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 2 3 4 Trifluoro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 5 Bromo 3 chloro 2 fluorophenylboronic acid 3 N N Dimethylamino phenylboronic acid pinacol ester 4 Chlorophenylboronic acid pinacol ester 4 Hydroxy 3 isopropylphenylboronic acid 3 5 Dimethyl 2 methoxyphenylboronic acid 2 Fluoro biphenyl 5 ylboronic acid 3 1H Tetrazol 5 yl phenyl boronic acid 5 Chloro 2 isopropoxypyridine 4 boronic acid 4 Methylbiphenyl 3 ylboronic acid 1 Methylindazole 5 boronic acid pinacol ester 3 Bromo 5 chloro 2 6 difluorophenylboronic acid 2 6 Difluoro 4 methylthio phenylboronic acid 2 6 Difluoro 3 methylthio phenylboronic acid pinacol ester 4 Pyridin 2 yl phenylboronic acid 4 Methoxy 2 methoxymethyl phenylboronic acid 2 5 Difluorophenylboronic acid pinacol ester 4 Formyl 2 trifluoromethyl phenylboronic acid pinacol ester 2 3 Dimethyl 4 methoxymethoxy phenylboronic acid 2 Chloro 4 trifluoromethyl phenylboronic acid pinacol ester 2 Chloro 6 trifluoromethyl phenylboronic acid pinacol ester 2 4 Bromo 2 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 Difluoro 3 propoxyphenylboronic acid 3 Ethoxy 2 6 difluorophenylboronic acid 4 Methoxy 3 methylthio phenylboronic acid 2 Choro 3 5 difluorophenylboronic acid 2 5 Difluoro 4 ethoxyphenylboronic acid

2 Methyl 6 methylthio 3 pyridylboronic acid 5 Chloro 2 methythio phenylboronic acid 5 Bromo 3 chloro 2 ethoxyphenylboronic acid 2 Fluoro 3 methoxypyridine 4 boronic acid 3 5 Difluoro 4 methylthio phenylboronic acid 2 Methoxy 4 methylthio pyridine 3 boronic acid 4 Methyl 2 methylthio 5 pyridylboronic acid 2 Fluoro 5 methylsulfanyl pyridin 3 yl boronic acid 5 Chloro 3 meththio phenylboronic acid 4 N O Dimethylhydroxylaminocarbonyl 2 chlorophenylboronic acid 20Chloro 4 1 piperidinylcarbonyl phenylboronic acid 2 Chloro 4 1 pyrrolidinylcarbonyl phenylboronic acid 2 Chloro 4 methylcarbamoyl phenylboronic acid 2 Isopropoxy 4 methylphenylboronic acid 4 Bromo 2 chloro 6 methylphenylboronic acid 4 Methyl 2 methylthio phenylboronic acid 2 Fluoro 3 methylsulfanyl phenylboronic acid 4 Methoxy 2 pyrrolidin 1 ylmethyl phenylboronic acid 6 Chloro 1H indazole 4 boronic acid pinacol ester 2 2 Methoxyethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 N N Diisopropylaminocarbonyl phenylboronic acid 3 Chloro 2 fluoropyridne 5 boronic acid 3 Methyl 2 methylthio pyridine 5 boronic acid 5 Methothio thiophene 2 boronic acid 3 Morpholinomethyl phenylboronic acid pinacol ester 4 Fluoro 3 methylthio phenylboronic acid 2 Dimethylamino 4 methylpyridine 5 boronic acid 5 Ethoxymethyl pyridine 3 boronic acid 2 Fluoro 5 isopropoxypyridine 3 boronic acid 3 Bromo 6 Chloro 2 fluorophenylboronic acid pinacol ester