1 Boc 3 isopropylpiperidine 3 carboxylic Acid 2 4 dimethoxy Benzenesulfonyl fluoride 2 3 fluoropyridin 2 yl oxy ethan 1 amine hydrochloride 2 3 difluoropyridine 4 carboxylic acid 2 fluoromethyl azetidine hydrochloride 3 trimethylsilyl ethynyl phenylboronic acid 3 3 difluorocyclopentan 1 amine hydrochloride 4 3 bromo 4 fluorophenyl 3 4 2 hydroxyethyl amino 1 2 5 oxadiazol 3 yl 4 5 dihydro 1 2 4 oxadiazol 5 one 3 fluoro 1H pyrrolo 2 3 b pyridine 6 carboxylic acid 5 trifluoromethyl pyrimidin 2 yl methanol 4 bromo 1 difluoromethyl 1H pyrazole 3 Oxo 3 4 dihydro 2H benzo b 1 4 oxazin 6 yl boronic acid 2 phenyl 1H pyrrole 3 bromothiophene 2 carbonitrile 2 5 chloro 2 2 methoxy 4 4 methylpiperazin 1 yl phenyl amino pyrimidin 4 yl amino N methylbenzenesulfonamide 4 bromo 2 carboxymethyl benzoic acid 2 fluoro 3 iodophenol 3 bromo 5 nitro 1H indazole 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 4 propoxyphenylboronic acid 2 chlorothiophene 3 carboxylic acid 6 fluoro 1 2 3 4 tetrahydroquinoline 3 4 Diaminoanisole dihydrochloride 1 3 Fluorophenyl ethanol 3 bromo 2 4 5 trifluoronitrobenzene 2 3 Dimethyl 4 nitroanisole 2 Fluoro 6 trifluoromethyl acetophenone 2 Chloro 5 iodonitrobenzene 3 5 Dimethylisoxazole 1 Bromo 4 difluoromethyl benzene

4 Fluoro 2 methyl 5 nitroacetophenone 4 Fluorocinnamaldehyde 2 4 Dimethylphenylhydrazine HCl 3 Bromo 5 chlorobenzonitrile 2 Methylbenzyl cyanide 3 4 5 Trifluorocinnamic acid 4 N boc amino phenylboronic acid pinacol ester 2 FLUORO 4 METHYLPHENOL 4 Bromo 3 5 dichloropyridine 4 Chloro 2 methylpyrimidine 5 Bromo 2 fluoroiodobenzene 2 Amino 4 6 dichloropyrimidine 5 carbaldehyde 2 Hydroxy 4 methoxyacetophenone 2 Bromo 4 fluorobenzyl bromide 1 2 Benzenedisulfonyl difluoride 6 Trifluoromethyl indoline 1 Boc 3 methoxy methyl carbamoyl piperidine 2 fluorocyclobutan 1 amine 3 3 difluorocyclopentan 1 amine 6 chloro 3 fluoro 1H pyrrolo 2 3 b pyridine 1 difluoromethyl 4 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 2 difluorobenzo d 1 3 dioxol 5 yl methanamine 4 tert butyl 2 chloroaniline 3 methyl 7 nitro 1H indazole 5 cyano 2 iodobenzoic acid 6 methoxypyridin 3 ol 3 amino 5 trifluoromethyl phenylboronic acid 3 5 dichloro 4 formylbenzoic acid 5 chloro 6 methylpyridin 3 ol 2 Fluoro 4 trifluoromethyl acetophenone

2 4 Diiodophenol 1 2 Diiodo 3 4 5 6 tetrafluorobenzene 1 3 5 Difluorophenyl ethanol 6 fluoro 3 4 dihydroquinolin 2 1H one 2 5 dibromothiophene 3 carboxylic acid 4 tert butoxycarbonylamino 3 methoxyphenylboronic acid 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 3 iodo 5 nitro 1H indazole 5 Chloro 2 fluoronitrobenzene 2 2 Dimethyl 5 hydroxymethyl 1 3 dixoane 5 Bromo 2 chlorobenzotrifluoride 5 Fluoro 2 methylacetophenone 2 Bromobenzene 1 3 dicarboxaldehyde 3 5 Difluorophenylhydrazine HCl 3 Methoxybenzyl cyanide 2 Bromo 5 chlorobenzonitrile 4 Methylcinnamic acid 2 FLUORO 4 METHOXYACETOPHENONE 4 Tert butyl 2 6 dinitroanisole 3 Bromo 2 cyano 5 chloropyridine 1S 2S N p tosyl 1 2 diphenylethylenediamine 2 6 Difluorobenzotrifluoride 3 4 Dihydro 2H pyran 1 2 Chloro 4 4 chlorophenoxy phenyl ethan 1 one 3 3 difluorocyclopentyl methanamine oxalic acid 3 3 difluoro 4 methylpiperidine hydrochloride 2 bromo 5 fluoropyridine 4 carbonitrile 2 fluorocyclobutyl methanol 1 Benzyl 3 aminopiperidine 3 nitro Benzenesulfonyl fluoride

6 Trifluoromethyl indole 3 fluoro 1H pyrrolo 2 3 b pyridin 4 amine 5 trifluoromethyl cyclohexane 1 3 dione 3 6 dichloro 4 trifluoromethyl pyridazine 4 Chloro 2 cyano 6 methylpyrimidine 5 bromo 6 methoxypyridin 3 ol 4 tert butyl 3 nitroaniline 4 formyl 3 methoxyphenylboronic acid 2 chloro 6 methoxy 4 trifluoromethyl pyridine 2 5 Difluorobenzeneethanol 4 Cyano 2 iodo N methylsulfonyl 5 trifluoromethyl aniline 2 chloro 5 hydroxyisonicotinaldehyde 2 bromothiophene 3 carboxylic acid 4 tert butoxycarbonylamino 3 fluorophenylboronic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 amine 4 bromomethyl 2 chlorooxazole 2 tert butyl 4 methylaniline 4 iodo 1 nitro 2 trifluoromethyl benzene 6 chloro 3 iodo 1H indazole 3 5 Difluoro 4 nitroanisole 2 6 bis trifluoromethyl bromobenzene 2 Fluoro 3 trifluoromethyl acetophenone 4 Methoxybenzyl 2 2 2 trichloroacetimidate 4 5 Dimethyl 1 3 dioxol 2 one 4 Chloro 2 fluoronitrobenzene 3 Bromo 5 chlorobenzotrifluoride 4 Fluoro 2 methylacetophenone 1 4 Benzenedicarboxaldehyde 2 5 Difluorophenylhydrazine HCl 3 Bromobenzonitrile