6 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 1 2 B PYRIDAZINE 3 4 BROMO PHENYL 3 FLUORO OXETANE 6 CHLORO 2 FLUOROPYRIDINE 3 CARBOXALDEHYDE 6 CHLORO 2 FLUORO 3 METHANESULFONYL PYRIDINE 6 CHLORO 2 FLUORO NICOTINIC ACID METHYL ESTER 4 CHLORO 2 FLUOROMETHYL PYRIMIDINE 1 6 CHLORO 2 METHYL PYRIDIN 3 YL 2 2 2 TRIFLUORO ETHANOL 2 TERT BUTOXYCARBONYLAMINO 4 4 4 TRIFLUORO 3 TRIFLUOROMETHYL BUTYRIC ACID 1 TRIFLUOROMETHYL CYCLOPROPANAMINE 5 FLUORO 2 METHOXYMETHYL PYRIMIDIN 4 OL 8 FLUORO 7 IODO 2 METHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID ETHYL ESTER 5 BROMO 2 TRIFLUOROMETHYL ISONICOTINIC ACID METHYL ESTER 5 7 DICHLORO 2 TRIFLUOROMETHYLPYRAZOLO 1 5 A PYRIMIDINE 5 7 DICHLORO 3 TRIFLUOROMETHYLPYRAZOLO 1 5 A PYRIMIDINE 8 8 DIMETHYL 3 TRIFLUOROMETHYL 5 6 7 8 TETRAHYDRO 1 6 NAPHTHYRIDINE 4 FLUORO 2 3 DIHYDRO 1H INDOLE 4 FLUORO 5 HYDROXY AZEPANE 1 CARBOXYLIC ACID TERT BUTYL ESTER 6 BROMO 5 4 FLUORO BENZENESULFONYL 1 3 DIHYDRO INDOL 2 ONE 4 METHYL 2 TRIFLUOROMETHYL THIAZOL 5 YL METHANOL 7 FLUORO PYRROLO 1 2 A QUINOXALINE 3 4 FLUORO BENZOYL PYRIDINE 2 CARBOXYLIC ACID 2 BROMO 4 TRIFLUOROMETHYL NICOTINIC ACID METHYL ESTER 6 BROMO 2 TRIFLUOROMETHYL NICOTINIC ACID METHYL ESTER 4 METHYL 1 5 TRIFLUOROMETHYL PYRIDIN 2 YL PYRROLIDINE 3 CARBOXYLIC ACID 8 FLUORO 2 METHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID 4 CHLORO 7 TRIFLUOROMETHOXY QUINAZOLINE 1 CARBOXYMETHYL 3 TRIFLUOROMETHYL 1 4 5 7 TETRAHYDRO PYRAZOLO 3 4 C PYRIDINE 6 CARBOXYLIC ACID TERT BUTYL ESTER 1 CHLORO 6 TRIFLUOROMETHYL ISOQUINOLINE 1 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDIN 3 YL ETHANONE 8 TRIFLUOROMETHYL H PYRROLO 1 2 A QUINOXALINE

5 CHLORO 7 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXYLIC ACID METHYL ESTER 2 2 difluoro 1 3 propanediol 1 3 cyclic sulfate 5 3 BENZYLOXYCARBONYLAMINO PYRROLIDIN 1 YL 4 FLUORO 1 METHYL 1H PYRAZOLE 3 CARBOXYLIC ACID ETHYL ESTER 7 FLUORO 2 3 DIHYDRO BENZOFURAN 4 OL 4 5 DIBROMO 2 TRIFLUOROMETHYL BENZONITRILE 4 CYCLOPROPYLMETHOXY 3 TRIFLUOROMETHYL PHENOL 4 BROMO 1 2 FLUOROPHENYL 3 METHYL 1H PYRAZOL 5 AMINE 3 AMINO 1 3 CHLORO 4 FLUORO BENZYL PYRROLIDIN 2 ONE 4 FLUORO 3 ISOPROPYL BENZYLAMINE 5 FLUORO 6 METHYL PYRIDINE 2 CARBOXYLIC ACID METHYL ESTER 2 BROMO 3 CHLORO 4 FLUORO 6 NITRO PHENOL 4 METHYL 2 TRIFLUOROMETHYL THIAZOLE 5 CARBOXYLIC ACID 4 FLUOROISOINDOLINE 3 fluoropiperidin 4 yl methanamine 4 fluoropiperidin 3 yl methanamine 1 benzyl 3 ethyl 4 4 difluoropiperidine 1 3 dicarboxylate 3 fluoro tetrahydro 2H pyran 4 ol 2 CHLORO 4 2 4 DIFLUORO PHENYL 6 7 DIHYDRO 5H 1 PYRINDINE 6 TRIFLUOROMETHYL PYRIDIN 2 YL METHANOL 2 CHLORO 6 FLUORO N HYDROXY BENZAMIDINE 7 4 FLUORO PHENYL 5 METHYL 4 OXO 4 5 DIHYDRO THIENO 3 4 C PYRIDINE 6 CARBOXYLIC ACID 1 BENZYL 4 TRIFLUOROMETHYL PYRROLIDINE 3 CARBOXYLIC ACID 3 BROMO 5 FLUORO 2 HYDROXYBENZALDEHYDE 4 4 difluorocyclohexyl methanol 5 4 FLUORO PHENYL 7 METHYL 8 OXO 7 8 DIHYDRO 1 7 NAPHTHYRIDINE 6 CARBALDEHYDE 1 PHENYLMETHYL 4 TRIFLUOROMETHYL TRANS 3 PYRROLIDINECARBOXYLIC ACID 9 4 4 aminopiperidin 1 yl butyl N 2 2 2 trifluoroethyl 9H fluorene 9 carboxamide 8 AMINO 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID ETHYL ESTER 1 BENZYL 3 TRIFLUOROMETHYL PYRROLIDINE 3 CARBOXYLIC ACID 6 CHLORO 3 TRIFLUOROMETHYL 1 2 4 TRIAZOLO 3 4 A PHTHALAZINE

1R 1 4 FLUOROPHENYL PROPYLAMINE 5 FLUORO 3 3 DIMETHYL 2 3 DIHYDRO 1H INDOLE 2S 4R 1 tert butyl 2 methyl 4 fluoropyrrolidine 1 2 dicarboxylate 1 BENZYL 3 TRIFLUOROMETHYL PYRROLIDIN 3 YL METHANOL 3 FLUOROSALICYLALDEHYDE 3 3 BROMO 4 FLUORO PHENYL 2 2 DIMETHYL CYCLOPROPANECARBOXYLIC ACID 5 FLUORO 3 METHYL BENZOFURAN 2 CHLORO 6 FLUORO 1 METHYL 1H BENZOIMIDAZOLE 4 5 6 7 TETRAHYDRO 3 TRIFLUOROMETHYL 1H INDAZOLE 4 1 1 2 2 2 PENTAFLUOROETHYL BENZOIC ACID 2 TERT BUTYL 4 FLUOROPHENOL 2 BROMO 1 2 METHYL 6 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDIN 3 YL ETHANONE 2 CHLORO 5 FLUORO 1 METHYL 1H BENZO D IMIDAZOLE 4 METHYL 2 4 TRIFLUOROMETHYL PHENYL PYRIDINE 2 2 difluoropropane 1 3 diol 5 TRIFLUOROMETHYL THIENO 3 2 B PYRIDINE 4 4 difluoropyrrolidine 2 carboxylic acid 3 AMINO 1 4 FLUOROBENZYL PYRROLIDIN 2 ONE 2 4 CHLOROPHENYL 2 2 DIFLUOROACETIC ACID 4 4 CHLORO BENZENESULFONYL 4 2 5 DIFLUORO PHENYL CYCLOHEXYLAMINE 2S 4S N TERT BUTOXYCARBONYL 4 TRIFLUOROMETHYLPROLINE 6 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 1 2 B PYRIDAZINE 3 SULFONIC ACID AMIDE 4 BROMO 1 4 FLUORO PHENYL 1H IMIDAZOLE 2S 4S methyl 4 fluoropyrrolidine 2 carboxylate hydrochloride 3 TRIFLUOROMETHYL 1H INDAZOLE 5 CHLORO 6 TRIFLUOROMETHYL NICOTINIC ACID 3 CHLORO 5 IODO 2 TRIFLUOROMETHYL PYRIDINE 3 CHLORO 2 TRIFLUOROMETHYL 4 PYRIDINECARBOXYLIC ACID 6 4 FLUORO PHENYL IMIDAZO2 1 BTHIAZOLE 2 4 FLUORO PHENYL 5 HYDROXY BENZOFURAN 3 CARBOXYLIC ACID ETHYL ESTER

3 fluoro tetrahydropyran 4 one 4 CHLOROMETHYL 2 4 FLUORO PHENYL 5 METHYL OXAZOLE 2 AMINO 4 4 4 TRIFLUORO BUTYRIC ACID ETHYL ESTER 5 CHLORO 3 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDIN 7 YL CARBAMIC ACID TERT BUTYL ESTER 3 4 FLUORO PHENYL 2 PYRIDIN 4 YL ACRYLONITRILE 3 3 DIFLUOROCYCLOBUTYL METHANOL 2 BROMO 3 IODO 6 TRIFLUOROMETHYL PYRIDINE 5 CHLORO 6 TRIFLUOROMETHYL PYRIDINE 2 CARBOXYLIC ACID 2 BROMO 6 TRIFLUOROMETHYL 3 TRIMETHYLSILANYL PYRIDINE 2 BROMO 4 TRIFLUOROMETHYL NICOTINIC ACID 6 CHLORO 5 FLUORO 3 METHYL BENZO B THIOPHENE 2 DIETHYLAMINO 5 2 2 2 TRIFLUORO ETHYL PYRIMIDIN 4 OL 1 4 FLUORO BENZYL 4 HYDROXY 1H PYRROLO 2 3 C PYRIDINE 5 CARBOXYLIC ACID METHYL ESTER 2 THIAZOLAMINE 4 5 FLUORO 1H PYRROLO 2 3 B PYRIDIN 3 YL 2 AMINO 6 FLUORO NICOTINAMIDE 5 FLUORO 3 3 DIMETHYL 1 3 DIHYDRO INDOL 2 ONE 1 BROMOMETHYL 3 TRIFLUOROMETHYLSULFONYL BENZENE 3 AMINO 4 FLUORO 6 MORPHOLIN 4 YL BENZO B THIOPHENE 2 CARBOXYLIC ACID AMIDE 3 CHLORO 5 FLUORO 2 HYDROXYBENZALDEHYDE 2 BROMOMETHYL 6 TRIFLUOROMETHYL PYRIDINE 6 7 DIMETHOXY 1 2 4 TRIFLUOROMETHYL PHENYL ETHYL 1 2 3 4 TETRAHYDRO ISOQUINOLINE 3 3 TRIFLUOROMETHYL PHENOXY AZETIDINE 4 FLUORO 3 ISOPROPYLBENZOIC ACID 2 BROMO 4 TRIFLUOROMETHYL BIPHENYL 4 YL ACETIC ACID METHYL ESTER 3 FLUORO 2 HYDROXY 6 METHYL BENZALDEHYDE 8 METHYL 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID 6 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 2 1 F PYRIDAZINE 3 CARBOXYLIC ACID 2 2 2 TRIFLUORO 1 2 4 6 TRICHLORO PHENYL ETHANONE 5 FLUORO 4 3 ISOPROPYL 2 METHYL 3H IMIDAZOL 4 YL PYRIMIDIN 2 YLAMINE 3 3 TRIFLUOROMETHYL PHENYL PIPERAZINE 1 CARBOXYLIC ACID TERT BUTYL ESTER