3 4 Fluorophenyl phenethyl alcohol 1 Methyl 2 methylthio 4 5 dihydro 1H imidazole hydroiodide 1 Methyl 4 nitroimidazole 6 Bromo N N dimethyl 2 quinazolinamine 1 Methyl 1H pyrazole 4 sulfonyl chloride 6 Chloro 4 pyridazinamine 6 Bromo 8 methoxyimidazo 1 2 a pyrazine 2 4 Dihydroxypteridine 2 3 Chloro 5 trifluoromethyl phenyl acetonitrile 4 Bromobenzo d isoxazole 7 Bromo 1 2 4 triazolo 1 5 a pyridin 2 amine 2 Methoxy 4 4 methylpiperazin 1 yl aniline 6 Bromo 3 iodoimidazo 1 2 a pyrazine 5 Ethynyl 3 methyl 1H indazole 4 Hydroxypyrimidine 5 carboxylic acid 2 5 6 Trichloro 4 methyl 3 pyridinecarbonitrile 2 4 Dichloro 5 7 dihydrofuro 3 4 d pyrimidine 4 Pyridin 3 yloxy benzoic acid 1R 4S 7 Boc 2 oxo 7 azabicyclo 2 2 1 heptane 3 Fluoropyrrolidine hydrochloride 2 Bromobenzo d thiazole 6 carbonitrile 3 Amino 6 chloro 2 pyrazinecarbonitrile 1 2 4 Triazolo 4 3 a pyrazine 3 carboxylic acid 4 Chloro 3 methyl 1H pyrrolo 2 3 b pyridine 1 Aminomethyl cyclobutanol 1 4 Bromophenyl cyclobutanamine hydrochloride 6 Bromoquinoline 4 carboxylic acid 6 Chloro 2 methyl 1H indole 6 Benzyloxy pyridine 2 carboxylic acid 6 Bromo 3 hydroxypicolinic acid

5 chloro 4 fluoro 2 nitrophenol 4 Benzyloxy 2 6 difluorophenylboronic acid 3 Amino 1H pyrazol 5 ol 1H pyrazolo 4 3 c pyridine 3 carboxylic acid 4 Chloro 6 isopropoxypyrimidine 7 Bromo 1 2 dihydroisoquinolin 3 4H one 1 Boc 3 iodo 1H indazole 5 Iodo 4 methylpyrimidine 2 Amino 4 morpholin 4 yl pyrimidine 2 Chloro 6 nitroquinoxaline 6 Bromo 1 2 4 triazolo 1 5 a pyrazine 8 Chloro 2 methylimidazo 1 2 a pyrazine 6 Chloro N methyl 5 nitro 4 pyrimidinamine 1 Boc 4 Cbz aminoazepane 3 Bromoimidazo 1 2 b pyridazin 6 ylamine 2 Methylsulfonyl pyrimidine 4 carboxylic acid 1 Boc 5 6 Dichloro 1H indole 6 8 Dibromo 1 2 4 triazolo 1 5 a pyrazine 5 Bromo 2 cyanobenzeneacetonitrile 2 4 Methylpiperazin 1 yl pyrimidin 5 amine 7 Bromothieno 2 3 b pyrazine 2 6 Dichloro 3 nitrobenzoic acid 3 Fluoro 4 methyl 5 hydroxybenzoic acid 4 3 Bromoimidazo 1 2 b pyridazin 6 yl morpholine 5 Amino 2 fluoro 4 nitrobenzotrifluoride 4 Bromo 2 chloro 3 fluorophenol 6 Bromo 1H indazole 4 carboxylic acid 3 tert butyl 1H pyrazol 4 carbaldehyde 3 3 Fluorophenoxy methyl piperidin 3 ol 7 Fluoroquinoline 6 carbaldehyde

4 Methyltetrahydro 2H pyran 4 ol 8 Bromoisoquinolin 1 2H one 5 Bromo 4 chloropyrimidin 2 amine 7 Bromoisoquinolin 3 amine 1 Pyridazin 4 yl ethanone 5 Ethynylpyrimidine 5 Bromo 3 fluoropyridin 2 amine 2 Amino 5 bromo 3 chloropyrazine 4 1 Piperazinyl 6 trifluoromethyl pyrimidine 4 Bromo 2 cyanobenzeneacetonitrile 2 Chlorothiazol 5 yl methylamine hydrochloride 7 Nitro 2 1H quinoxalinone 5 Bromo 2 chlorobenzyl amine 3 5 Dimethylpyrazin 2 ol 7 Fluoro 1H indole 2 carboxylic acid 2 hydroxy 4 methylthiazole 5 carboxylicacid 5 Chloro 1 3 4 thiadiazol 2 amine 5 Bromo N methylpyrimidin 4 amine 4 5 Dichloropyrimidin 2 amine 5 Methyl 3 nitro 1H pyrazole 4 Flurophenyl acetic acid ethyl ester 2 3 4 5 Tetrahydro 1H benzo c azepine hydrochloride 2 3 Dibromopyrazine 1R 2S 2 Aminocyclohexanol hydrochloride 4 1 Pyrrolidinyl 3 trifluoromethyl bezenamine dihydrochloride 4 2 Bromoethyl benzonitrile 2 2 4 Dichlorophenyl thiazole 4 carboxylic acid 3 Phenyl 3 pentylamine hydrochloride 3 Amino 2 fluorophenyl methanol 2 4 Dichloro 5 6 7 8 tetrahydropyrido 4 3 d pyrimidine hydrochloride

1 2 3 4 Tetrahydropyrido 2 3 b pyrazine 2 Amino 3 methoxybenzaldehyde 4 Chloro 6 trifluoromethyl 1H pyrazolo 3 4 d pyrimidine 6 Bromochromen 2 one 2 Chloro 4 morpholinothieno 3 2 d pyrimidine 6 carbaldehyde 4 Amino N methylbenzeneethanesulfonamide 1 Piperidin 4 yl pyrrolidin 2 one 2 Chloro 5 isopropylpyrimidine 4 Amino 6 iodopyrimidine 4 Chloro 7 trifluoromethyl quinazoline 4 Methylamino 3 nitropyridine 6 Hydroxyimidazo 1 2 b pyridazine 1 Boc 3 Cyano 4 hydroxypyrrolidine 1 Boc 3 Iodo 7 azaindole 2 4 Methyl 1 piperazinyl 4 pyrimidinamine 2 Amino 6 bromopyrido 2 3 d pyrimidin 4 3H one 3 4 Bromopyrazol 1 ylmethyl pyridine 6 Hydroxy 1 2 benzisoxazole 1 Boc 5 Bromo 1 2 dihydro 2 oxo spiro 3H indole 3 4 piperidine 2 4 Bromo 1H pyrazol 1 yl pyrimidine 2 Methylsulfonyl 5 bromopyrimidine 4 carboxylic acid 1 Boc 4 4 Benzylpiperazin 1 yl 4 methylpiperidine 4 Chloro 6 7 dimethylenedioxyquinazoline 2 3 5 Dichlorophenyl thiazole 4 carboxylic acid 2 4 Diiodopyrimidine 4 5 Bromopyrimidin 2 yloxy phenyl methanol 5 Bromo 2 3 methoxypropylamino pyrimidine 2 4 Nitrophenoxy pyrimidine 5 Bromo 2 4 nitrophenoxy pyrimidine 1 5 Bromopyrimidin 2 yl piperidin 3 yl methanol