2 Bromo 5 methylthiopyridine 6 Fluoro 2 methylpyridine 3 carboxaldehyde 5 Bromo 3 methyl N cyclohexylpyridine 2 carboxamide 5 Bromo 3 methyl 2 piperidin 1 yl carbonyl pyridine 5 Bromo 3 methylpyridine 2 carbonyl chloride 2 Benzyloxy 5 bromo 4 methylpyridine 3 Bromo 2 chloro 4 iodopyridine 5 Chloro 2 propan 2 yloxy pyridine 4 Benzyloxy 1 3 dibromobenzene 5 Bromo 2 fluoro 3 methylbenzaldehyde 4 Bromo 2 6 dichloro ethoxybenzene 3 5 Dichloro 4 benzyloxybromobenzene 6 Chloro 2 fluoro 3 methoxybenzaldehyde 2 Chloro 6 fluoro 3 methylbenzaldehyde 3 Bromo 2 chloro 6 fluorobenzaldehyde 2 Chloro 6 fluoro 3 methoxybenzoic acid 2 3 Dichloro 6 fluorobenzaldehyde 2 3 Dichloro 6 fluorobenzoic acid 2 6 Dibromo 4 fluoroanisole 3 Bromo 6 chloro 2 fluorobenzaldehyde 3 Benzyloxy 6 bromo 2 fluorobenzaldehyde 6 Bromo 3 ethoxy 2 fluorobenzaldehyde 5 Bromo N tert butylnicotinamide 1 Benzyloxy 2 Bromo 4 trifluoromethylbenzene 2 Chloro 3 hydroxybenzotrifluoride 2 Fluoro 3 methyl pyridine 5 carboxylic acid 6 Chloro 5 methylpyridine 3 carbaldehyde 2 Chloro 3 fluoro 5 iodopyridine 6 Bromo 8 methylimidazo 1 2 a pyridine 6 Bromoimidazo 1 2 a pyridine hydrochloride

2 5 Dibromonicotinaldehyde 2 Bromo 3 methylpyridine 5 carboxylic acid 2 6 Dimethoxypyridine 3 carboxaldehyde 4 Bromo 2 fluoro 3 methylpyridine 4 Bromo 2 chloro 3 iodopyridine 5 Bromo 2 fluoro 3 methoxypyridine 5 Fluoropyridin 3 yl methanol 5 Bromo 2 pyrrolindin 1 ylcarbonyl pyridine 5 Bromopyridine 2 yl morpholino methanone 5 Bromo N N dimethyl 3 pyridinecarboxamide 5 Bromo methyl 3 pyridinecarboxamide 5 Bromo 3 pyrrolidin 1 ylcarbonyl pyridine 5 Bromo 3 piperidin 1 ylcarbonyl pyridine 5 Chloro 2 methylthiopyridine 5 Bromo 2 piperidin 1 ylcarbonyl pyridine 5 Bromopyridine 2 carboxylic acid diethylamide 2 Methylbiphenyl 4 ylboronic acid 3 Bromo 5 trifluoromethoxy phenylboronic acid pinacol ester 2 6 Difluoro 4 hydroxyphenylboronic acid pinacol ester 2 4 Difluoro 5 methoxyphenylboronic acid pinacol ester 2 4 Difluoro 5 methoxyphenylboronic acid 6 Chloro 5 methoxypyridine 3 boronic acid pinacol ester 3 Fluoro 5 hydroxymethyl phenylboronic acid pinacol ester 2 4 Dichloro 3 methoxyphenylboronic acid pinacol ester 3 Iodophenylboronic acid pinacol ester 4 Acetyl 3 fluorophenylboronic acid pinacol ester 2 Methoxy 1 naphthaleneboronic acid pinacol ester 4 Chloro 3 fluoro 2 formylphenylboronic acid pinacol ester 4 Hydroxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 4 Ethoxycarbonyl 3 fluorophenylboronic acid pinacol ester

4 Chloro 3 hydroxymethyl phenylboronic acid pinacol ester 4 Bromo 2 5 dimethylphenylboronic acid pinacol ester 2 Trifluoromethyl phenylboronic acid pinacol ester 2 Fluoro 4 formylphenylboronic acid pinacol ester 1 Propylboronic acid pinacol ester 2 3 Bromo 5 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Methoxy 5 trifluoromethyl phenylboronic acidpinacol ester 2 Fluoro 3 trifluoromethyl phenylboronic acid pinacol ester 2 Fluoro 4 methylthiophenylboronic acid pinacol ester 4 Isopropyl 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 3 Bromo 5 methoxyphenylboronic acid pinacol ester 3 Bromo 5 ethoxyphenylboronic acid pinacol ester 5 Chloro 2 pivaloylamino phenylboronic acid pinacol ester 5 Methothio thiophene 2 boronic acid pinacol ester 4 Chloro 3 fluorophenylboronic acid pinacol ester 2 2 3 Dimethoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Hydroxymethyl 4 methylphenylboronic acid pinacol ester 4 Piperidin 1 ylmethyl phenylboronic acid pinacol ester 3 Chloro 4 isopropoxyphenylboronic acid pinacol ester 4 Cyclohexylaminocarbonyl phenylboronic acid pinacol ester 2 Fluoro 6 methoxyphenylboronic acid pinacol ester 2 6 Dichlorophenylboronic acid pinacol ester 2 Formyl 4 trifluoromethyl phenylboronic acid pinacol ester 5 Chloro 2 isopropoxypyridine 3 boronic acid 2 4 Bromo 3 5 dichlorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 5 Isopropoxy 2 methylphenylboronic acid pinacol ester 2 Chloro 6 trifluoromethyl pyridine 4 boronic acid 1 3 Bis 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzene 3 Isopropylphenylboronic acid pinacol ester 2 3 Dichloropyridine 5 boronic acid

4 Benzyloxy 2 methoxyphenylboronic acid pinacol ester 3 Bromo 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 2 2 Methoxy 4 5 dimethylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 2 Morpholinoethoxy phenylboronic acid HCl 4 Isopropoxy 3 methoxyphenylboronic acid pinacol ester 1 trifluoromethyl 1H pyrazole 4 boronic acid pinacol ester 3 5 Dimethyl 4 isopropoxyphenylboronic acid 2 Chloro 4 5 difluorophenylboronic acid 4 4 Methylpiperazine 1 carbonyl phenylboronic acid pinacol ester 4 4 Methylpiperazine 1 carbonyl phenylboronic acid 4 Benzyloxy 2 trifluoromethylphenylboronic acid pinacol ester 4 Benzyloxy 2 trifluoromethoxy phenylboronic acid 3 Bromo 4 methoxyphenylboronic acid pinacol ester 3 Bromo 4 fluorophenylboronic acid pinacol ester 5 4 Morpholinylmethyl thiophene 2 boronic acid pinacol ester 3 Hydroxy 2 methylphenylboronic acid 2 Methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 3 Cyclobutylphenylboronic acid 2 5 Difluoro 6 methylbenzeneboronic acid pinacol ester 4 Cyano 3 ethylphenylboronic acid 2 6 Dimethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 2 Bromo 5 trifluoromethylphenylboronic acid pinacol ester 3 Methoxy 4 phenoxyphenylboronic acid 4 Cyclobutylphenyl boronic acid 5 Butylthiophen 2 boronic acid 5 Bromo 2 fluorophenylboronic acid pinacol ester 4 Fluorobenzofuran 7 boronic acid 2 2 5 bis Trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 Bromo 5 chlorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 Bis trifluoromethyl phenylboronic acid pinacol ester