6 fluoro 1H pyrrolo 2 3 b pyridin 4 amine 4 azetidin 3 yl 2 2 dimethylmorpholine bis trifluoroacetic acid 2 tert butoxy carbonyl 5 5 difluoro octahydrocyclopenta c pyrrole 1 carboxylic acid 2 fluoropyridin 3 yl 3 hydroxypiperidin 1 yl methanone 4 Fluoro 1H benzimidazole 2 5 dibromo 4 iodopyridine 6 bromo 3 methylquinazolin 4 3H one 1 4 chlorophenyl N 3 cyano 4 4 morpholinopiperidin 1 yl phenyl 5 methyl 1H pyrazole 4 carboxamide 4 borono 2 nitrobenzoic acid 3 amino 6 trifluoromethyl pyridin 2 ol 2 3 dihydrobenzofuran 5 amine 2 bromo 4 methoxy 1 trifluoromethyl benzene 3 methoxy 2 nitroaniline 7 bromo 3 chloro 1H indazole 1H indazol 6 yl boronic acid 2 methylimidazo 1 2 a pyridine 3 carbaldehyde 3 Fluoro 4 trifluoromethyl benzoic aicd 2 3 5 6 Tetrafluorobenzyl bromide 2 3 Difluoro 5 nitroacetophenone 2 5 Dibromophenol 2 4 6 Trichlorobromobenzene 2 3 5 Trifluorobenzoic acid 5 Bromo 2 4 difluoronitrobenzene 4 Chloromethyl 3 5 dimethylisoxazole 4 Nitrobenzaldehyde 4 Ethoxyacetophenone 2 Amino 5 chloro 3 iodobenzonitrile 3 4 Trifluoromethoxy phenyl propanoic acid 4 BROMO 2 3 DICHLOROANILINE 3 Fluoro 2 iodobenzaldehyde

2 4 Amino 1 tert butoxycarbonyl piperidin 4 yl acetic acid 4 4 Bromophenyl piperidine 4 Hydroxy 3 nitropyridine 5 Bromo 2 iodo 1 3 dimethylbenzene 2 Fluoro 5 iodobenzonitrile 4 tert butyl 2 chloropyridine 6 Bromoindole 2 6 Dimethyl 4 Hydroxybenzaldehyde 3 2 4 5 trifluorophenyl azetidin 3 ol 1 N Boc aminomethyl 4 aminomethyl benzene 6H Pyrimido 5 4 b 1 4 oxazin 7 8H one 2 trans 4 1R 1 amino 2 7 fluoro 2 oxo 1 2H quinoxalinyl ethyl cyclohexyl amino methyl 2 2 difluoro 3 methoxypropanoic acid 4 bromo 6 fluoro 1H pyrrolo 2 3 b pyridine 1 2 amino 5 bromophenyl propan 1 one 4 chloro 2 cyanophenylboronic acid 3 2 cyanopropan 2 yl N 4 methyl 3 3 methyl 4 oxo 3 4 dihydroquinazolin 6 ylamino phenyl benzamide 4 Quinolinemethanamine hydrochloride 1 1 3 chloro 2 nitrophenol 5 chloro 2 fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 chloropyridin 3 amine 3 bromo 4 5 dihydroxybenzaldehyde 3 bromo 5 nitrophenol 4 fluoro 3 iodo 1H indazole 1H indazol 7 yl boronic acid 2 3 dimethylimidazo 1 2 a pyridine 7 carbaldehyde 4 Propylbenzyl bromide 3 4 5 Trichlorobenzoic acid 2 3 4 6 Tetramethyl 1 fluorobenzene 4 Ethoxybenzol 1 2 diamin 2 6 Dichloro 4 trifluoromethyl acetophenone

5 Chlorofuran 2 carboxylic acid 5 Bromo 2 3 difluoronitrobenzene 4 Trifluoromethyl thiophenol 3 5 Dimethyl 2 hydroxyacetophenone 3 Nitrobenzaldehyde 3 Methoxyphenethylamine 3 5 Dichlorobenzyl cyanide 5 Amino 2 chlorobenzonitrile 3 3 Nitrophenyl propanoic acid 2 3 5 6 Tetrachloro 1 4 dicarboxylic acid 1 BROMO 2 5 DICHLOROBENZENE 2 Isopropoxy 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 Difluorophenylhydrazine hydrochloride 6 Benzylaminopurine 3 4 Boc piperazin 1 yl aniline 3 Hydroxy thiophenol 3 Amino 4 fluorophenol 3 Methylbenzotrifluoride 2 3 5 Triiodobenzoic acid 1 4 FLUORO PHENYL CYCLOPROPANECARBOXYLIC ACID 3 2 3 5 trifluorophenyl azetidin 3 ol 3S 4R 4 fluoropyrrolidin 3 ol hydrochloride 4 chloro 6 fluoro 1H pyrrolo 2 3 b pyridine 2 Isopropylpyridin 3 amine 1 2 dihydrospiro indole 3 4 piperidine 2 one trifluoroacetic acid 1 trifluoromethyl cyclopropyl methanamine hydrochloride 4 fluoro 3 3 dimethylindoline 6 chlorobenzo b thiophene 2 carboxylic acid 7 methyl 1 5 dioxo 1 2 3 5 tetrahydroindolizine 6 carbonitrile 3 benzyloxy 4 methoxyphenylboronic acid

1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl indolin 1 yl ethanone 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 7 trifluoromethyl 1H indazole 7 methylimidazo 1 2 a pyrimidine 3 carbaldehyde 5 bromo 2 tert butyl pyrimidine 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 3 trifluoromethyl pyridine 1 2 chloro 5 trifluoromethyl pyridin 3 yl ethanone 3 4 dibromophenol 3 bromo 4 fluoro 1H indazole 4 propylbenzyl alcohol 2 3 Chloropropyl 2 4 fluorophenyl 1 3 dioxolane 3 5 Dichloro 2 2 2 trifluoroacetophenone 4 Methoxy 1 2 phenylenediamine 2 3 5 6 Tetrafluorobenzoic acid 2 3 5 6 Tetrafluoronitrobenzene 2 4 Dichloro 5 fluoro 3 nitrobenzoic acid 5 Bromo 2 thiophenemethanamine 3 4 Methylenedioxy phenylpropionic acid 4 Nitrobenzene 1 2 dicarboxylic acid 4 Amino 3 chlorobenzonitrile 2 6 Dichlorobenzyl cyanide 4 Fluorophenethylamine 4 Methylsulfonyl 2 trifluoromethyl benzaldehyde 4 Dimethylaminoacetophenone 3 Trifluoromethyl thiophenol 4 Bromo 2 6 difluoronitrobenzene 2 bromo 5 fluoroaniline hydrochloride 2 4 Dibromo 3 fluoroaniline 5 Bromofuran 2 carbonyl chloride 4 Methoxythiophenol 6 Dimethylaminopurine