1 4 Chloro 3 nitrobenzenesulfonyl 1 2 3 4 tetrahydroquinoline 4 Chloro 6 pyrrolidin 1 yl 2 trifluoromethylpyrimidine 5 4 Fluorophenyl pyridine 2 carbonitrile 7 Benzyloxyindol 1 yl acetic acid 1 Boc 2 3 Bromophenyl piperazine 2 2 Fluorophenyl pyrimidine 5 carbaldehyde 5 m Tolyl pyridin 2 amine dihydrochloride 1 Bis 4 fluorophenyl methyl 4 4 nitrophenyl piperazine 4 4 Bis 4 fluorophenyl methyl piperazin 1 yl phenylamine 3 4 Methoxyphenyl thiomorpholine 2 2 5 Dimethoxyphenyl piperazine 4 2 Methylimidazol 1 ylmethyl phenylamine 3 3 Bromo 4 methoxyphenyl pyridine 1 Boc 4 2 Carboxybenzyl piperazine 2 2 Methylimidazol 1 yl phenyl methanol 2 1 2 4 Triazol 1 yl phenyl methanol 3 6 Chloropyridazin 3 yl benzoic acid 5 2 5 Dimethoxyphenyl 1H pyrazole 3 carboxylic acid 1 Pyridin 2 ylmethylpiperidin 4 yl methanol 1 4 Hydroxymethylphenyl piperidin 4 ol 1 Boc 3 Hydroxymethyl 7 nitroindole 1 Boc 3 Hydroxymethyl 7 methylindole 1 Boc 3 Hydroxymethyl 6 methoxyindole 1 Boc 5 Bromo 3 hydroxymethylindole 1 Boc 4 Bromo 3 hydroxymethylindole 1 Boc 3 Hydroxymethyl 6 methylindole 1 Boc 3 Hydroxymethyl 5 methylindole 1 Boc 4 Chloro 3 hydroxymethylindole 1 Boc 4 Chloro 3 formylindole 2 6 Methoxynaphthalen 2 yl piperazine

2 2 5 Dichlorophenyl piperazine 1 Boc 5 Methyl 3 formylindole 1 Boc 6 Methyl 3 formylindole 1 Boc 7 Methyl 3 formylindole 2 3 5 Dimethoxyphenyl piperazine 4 Chloro 2 2 benzoxazolylthio 5 thiazolecarboxaldehyde 2 4 Bromophenyl thiazole 5 carbaldehyde 2 4 Fluorophenyl thiazole 5 carbaldehyde 2 3 Fluorophenyl thiazole 5 carbaldehyde 4 Methyl 1 4 amino 2 trifluoromethylphenyl piperidine dihydrochloride 1 5 Chloro 1H indazol 1 yl ethanone 5 Bromo 1 3 di tert butyl 2 methoxybenzene 4 Bromo 2 methyl 1H pyrrolo 2 3 b pyridine 4 Dibenzylamino cyclohexanone 6 Fluorobenzo d isoxazol 3 amine 5 Pyrimidineethanol 2 Amino 4 5 Difluorophenol 6 Bromoimidazo 1 2 a pyrazine 3 carbaldehyde 6 Benzyl 6 7 dihydro 1H pyrrolo 3 4 d pyrimidine 2 4 3H 5H dione 6 Amino 7 bromobenzothiazole 5 Trifluoromethyl 1H pyrrolo 2 3 b pyridine 5 Bromo 4 chloro 6 methylpyrimidine 5 Bromo 3 ethynylpyridin 2 ylamine 5 Bromo 2 chloro 7H pyrrolo 2 3 d pyrimidine 5 Bromo 1H 1 2 4 triazole 3 carboxylic acid 5 Aminopyridin 3 ol dihydrochloride 5 Trifluoromethyl 1H pyrazole 4 carboxylic acid 4 Chlorobenzothiazole 4 Chloro 7H pyrrolo 2 3 d pyrimidine 5 carboxylic acid 4 Chloro 7H pyrrolo 2 3 d pyrimidine 5 carbonitrile

4 Bromoquinoline 6 carboxylic acid 7 tert Butyl 3 ethyl 5 6 dihydro 1 2 4 triazolo 4 3 a pyrazine 3 7 8H dicarboxylate 8 Bromo 2H 1 benzopyran 2 one 6 Methyl 2 4 dihydroxyquinoline 6 Bromo 4 chloropyrido 2 3 d pyrimidine 1 5 Bromothiophen 3 yl ethanone 4 Phenoxy 6 chloropyrimidine 4 Chloro 7H pyrrolo 2 3 d pyrimidine 6 carboxylic acid 5 Bromo 2 phenyl 1H pyrrolo 2 3 b pyridine 5 Bromo 2 methoxypyrimidin 4 ylamine 3 Chloro 5 Nitropyridine 4 amine 2 Hydroxy 5 methylpyrazine 3 Chloro 2 methoxybenzaldehyde 4 Bromo 2 methylisoquinolin 1 2H one 3 5 Dibromo N N dimethylpyrazinamine 3 Amino 1 cyclopentyl 1H pyrazole 4 carbonitrile 4 Bromo 1 methoxyisoquinoline 2 Hydroxy 3 6 dimethylbenzaldehyde 2 Methyl 2H indazol 4 amine 2 tert Butoxycarbonylaminomalonic acid monoethyl ester 2 Chloro 6 fluoroquinoxaline 2 Chloro 5 iodopyrazine 2 Bromo 6 methylpyrazino 2 3 b pyrazine 2 Bromo 4 5 6 7 tetrahydrothiazolo 5 4 c pyridine hydrochloride 2 Amino N N diethylbenzenesulfonamide 2 Amino 6 cyanopyrazine 1 Boc 5 Chloro 6 trifluoromethyl 1H indole 2 3 Dihydro 2 phenyl 4 1H quinolinone 2 6 Dibromoquinazoline 2 Amino 5 iodopyrazine

2 Amino 6 bromopyrazine 1 Boc 5 6 Dichloro 1H indole 2 boronic acid 2 Aminomethyl benzonitrile 6 Chloro 1 2 3 4 tetrahydropyrido 2 3 b pyrazine 6 Bromo 2 methylisoquinolin 1 2H one 2 4 2 Aminobenzenesulfonyl piperazin 1 yl ethanol 2 Iodobenzothiazole 1 Tosyl 1H pyrrolo 2 3 b pyridin 3 ylboronic acid 1 Boc 1 2 dihydro 5 methoxy 2 oxo spiro 3H indole 3 4 piperidine 6 Chloro 5 nitroquinoline 5 Bromopyridin 2 yl methyl carbamic acid tert butyl ester 3 Iodopicolinic acid 3 Methoxy 4 methyl 2 nitrobenzoic acid 4 Imidazo 1 2 a pyrazin 2 yl 1 2 5 oxadiazol 3 amine 1 Boc 5 Fluoro 1 2 dihydro 2 oxo spiro 3H indole 3 4 piperidine 1 Boc 4 4 Bromo 2 formylphenyl piperazine 1 4 Piperidinyl 2 trifluoromethyl 1H benzimidazole 1H Indazole 7 carboxamide 1 Phenylsulfonyl 1H pyrrolo 2 3 b pyridine 4 Bromothiazol 5 yl methanol 1 Methyl 1H pyrazol 4 amine hydrochloride 1 3 Benzodioxole 4 carbonylchloride 2 Amino 4 iodopyrimidine 2 Chloro 6 nitroquinoline 6 Bromo 8 chloroimidazo 1 2 a pyrazine 3 3 Dimethylpiperidin 4 ol 2 4 Iodophenyl ethanol 2 4 Dibromothiazol 5 yl methanol 1 Boc pyrazole 5 Methyl 2 piperazin 1 yl thiazole