1 Boc 4 2 Carboxybenzyl piperazine 3 3 Bromo 4 methoxyphenyl pyridine 2 1 2 4 Triazol 1 yl phenyl methanol 3 6 Chloropyridazin 3 yl benzoic acid 2 2 Methylimidazol 1 yl phenyl methanol 5 2 5 Dimethoxyphenyl 1H pyrazole 3 carboxylic acid 1 Boc 3 Hydroxymethyl 7 nitroindole 1 4 Hydroxymethylphenyl piperidin 4 ol 1 Boc 3 Hydroxymethyl 6 methoxyindole 1 Pyridin 2 ylmethylpiperidin 4 yl methanol 1 Boc 3 Hydroxymethyl 7 methylindole 1 Boc 5 Bromo 3 hydroxymethylindole 1 Boc 4 Bromo 3 hydroxymethylindole 1 Boc 3 Hydroxymethyl 6 methylindole 1 Boc 3 Hydroxymethyl 5 methylindole 1 Boc 4 Chloro 3 formylindole 1 Boc 4 Chloro 3 hydroxymethylindole 1 Boc 5 Methyl 3 formylindole 1 Boc 6 Methyl 3 formylindole 1 Boc 7 Methyl 3 formylindole 2 2 5 Dichlorophenyl piperazine 2 6 Methoxynaphthalen 2 yl piperazine 2 3 5 Dimethoxyphenyl piperazine 4 Methyl 1 4 amino 2 trifluoromethylphenyl piperidine dihydrochloride 4 Chloro 2 2 benzoxazolylthio 5 thiazolecarboxaldehyde 2 4 Bromophenyl thiazole 5 carbaldehyde 2 4 Fluorophenyl thiazole 5 carbaldehyde 2 3 Fluorophenyl thiazole 5 carbaldehyde 4 Dibenzylamino cyclohexanone 1 5 Chloro 1H indazol 1 yl ethanone

5 Bromo 1 3 di tert butyl 2 methoxybenzene 4 Bromo 2 methyl 1H pyrrolo 2 3 b pyridine 2 Amino 4 5 Difluorophenol 5 Pyrimidineethanol 5 Trifluoromethyl 1H pyrrolo 2 3 b pyridine 6 Amino 7 bromobenzothiazole 6 Benzyl 6 7 dihydro 1H pyrrolo 3 4 d pyrimidine 2 4 3H 5H dione 6 Bromoimidazo 1 2 a pyrazine 3 carbaldehyde 6 Fluorobenzo d isoxazol 3 amine 5 Bromo 4 chloro 6 methylpyrimidine 5 Bromo 3 ethynylpyridin 2 ylamine 5 Bromo 2 chloro 7H pyrrolo 2 3 d pyrimidine 5 Bromo 1H 1 2 4 triazole 3 carboxylic acid 5 Aminopyridin 3 ol dihydrochloride 5 Trifluoromethyl 1H pyrazole 4 carboxylic acid 4 Chlorobenzothiazole 4 Chloro 7H pyrrolo 2 3 d pyrimidine 5 carboxylic acid 4 Chloro 7H pyrrolo 2 3 d pyrimidine 5 carbonitrile 4 Bromoquinoline 6 carboxylic acid 8 Bromo 2H 1 benzopyran 2 one 6 Methyl 2 4 dihydroxyquinoline 7 tert Butyl 3 ethyl 5 6 dihydro 1 2 4 triazolo 4 3 a pyrazine 3 7 8H dicarboxylate 6 Bromo 4 chloropyrido 2 3 d pyrimidine 1 5 Bromothiophen 3 yl ethanone 4 Phenoxy 6 chloropyrimidine 4 Chloro 7H pyrrolo 2 3 d pyrimidine 6 carboxylic acid 2 Hydroxy 5 methylpyrazine 3 Chloro 5 Nitropyridine 4 amine 5 Bromo 2 phenyl 1H pyrrolo 2 3 b pyridine 5 Bromo 2 methoxypyrimidin 4 ylamine

3 5 Dibromo N N dimethylpyrazinamine 3 Amino 1 cyclopentyl 1H pyrazole 4 carbonitrile 3 Chloro 2 methoxybenzaldehyde 4 Bromo 2 methylisoquinolin 1 2H one 4 Bromo 1 methoxyisoquinoline 2 Methyl 2H indazol 4 amine 2 tert Butoxycarbonylaminomalonic acid monoethyl ester 2 Bromo 6 methylpyrazino 2 3 b pyrazine 2 Chloro 5 iodopyrazine 2 Chloro 6 fluoroquinoxaline 2 Hydroxy 3 6 dimethylbenzaldehyde 2 Amino N N diethylbenzenesulfonamide 2 Bromo 4 5 6 7 tetrahydrothiazolo 5 4 c pyridine hydrochloride 2 6 Dibromoquinazoline 2 Amino 5 iodopyrazine 2 Amino 6 bromopyrazine 2 Amino 6 cyanopyrazine 2 3 Dihydro 2 phenyl 4 1H quinolinone 1 Boc 5 6 Dichloro 1H indole 2 boronic acid 1 Boc 5 Chloro 6 trifluoromethyl 1H indole 2 Iodobenzothiazole 6 Bromo 2 methylisoquinolin 1 2H one 6 Chloro 1 2 3 4 tetrahydropyrido 2 3 b pyrazine 2 Aminomethyl benzonitrile 2 4 2 Aminobenzenesulfonyl piperazin 1 yl ethanol 1 Boc 1 2 dihydro 5 methoxy 2 oxo spiro 3H indole 3 4 piperidine 5 Bromopyridin 2 yl methyl carbamic acid tert butyl ester 6 Chloro 5 nitroquinoline 3 Iodopicolinic acid 1H Indazole 7 carboxamide

3 Methoxy 4 methyl 2 nitrobenzoic acid 4 Imidazo 1 2 a pyrazin 2 yl 1 2 5 oxadiazol 3 amine 1 Tosyl 1H pyrrolo 2 3 b pyridin 3 ylboronic acid 1 Boc 5 Fluoro 1 2 dihydro 2 oxo spiro 3H indole 3 4 piperidine 1 Boc 4 4 Bromo 2 formylphenyl piperazine 1 4 Piperidinyl 2 trifluoromethyl 1H benzimidazole 1 Phenylsulfonyl 1H pyrrolo 2 3 b pyridine 4 Bromothiazol 5 yl methanol 1 Methyl 1H pyrazol 4 amine hydrochloride 1 3 Benzodioxole 4 carbonylchloride 6 Bromo 8 chloroimidazo 1 2 a pyrazine 2 Chloro 6 nitroquinoline 2 Amino 4 iodopyrimidine 3 3 Dimethylpiperidin 4 ol 2 4 Iodophenyl ethanol 2 4 Dibromothiazol 5 yl methanol 1 Boc pyrazole 4 Chloro 5 fluoropyrimidine 5 Methyl 2 piperazin 1 yl thiazole 7 Amino N methyl 1 2 3 4 tetrahydroquinoline hydrochloride 1 5 Bromopyridin 3 yl N methylmethanamine 1 Boc 3 bromopyrrolidine 3 Aminophenylacetic acid methyl ester 4 Nitroisoxazole 6 Chloro 2 methylimidazo 1 2 b pyridazine 3 carboxylic acid 2 3 4 Dichlorophenyl 1 2 pyrrolidin 1 ylmethyl piperidin 1 yl ethanone hydrochloride 3beta 20beta 3 3 Carboxy 1 oxopropoxy 11 oxoolean 12 en 29 oic acid 6 Chloro 3 nitroimidazo 1 2 b pyridazine 6 Chloro 3 hydroxypyridazine 4 carboxylic acid 6 Chloroimidazo 1 2 b pyridazin 3 ylamine