2 Amino 3 iodo 6 methylpyridine 2 Bromo 5 trifluoromethoxy aniline 2 Chlorobenzimidazole 2 4 Dibromopyridine 3 fluoropyrazine 2 carboxylic acid 3 1 fluoroethyl azetidine 4 Methyl 2 oxopentanoic acid methyl ester 3 4 5 triethoxybenzoic acid 2 Bromo 6 picoline 2 Bromo 5 nitrobenzoic acid 3 Fluoropyridin 4 yl boronic acid 5 chloro 6 fluoro 1H indole 2‐ tert‐butoxy carbonyl amino ‐3‐ 3 3‐difluorocyclobutyl propanoic acid 3 5 difluoro 4 4 4 fluorophenyl piperidin 1 yl aniline 2 4 trifluoromethyl phenyl piperazine dihydrochloride 3 fluorooxetan 3 yl methanol 2R 3R 4R 5R 5 2 amino 6 chloro 9H purin 9 yl 2 4 chlorobenzoyloxy methyl 4 fluoro 4 methyloxolan 3 yl 4 chlorobenzoate 1 tert butoxycarbonyl 2 oxospiro indoline 3 4 piperidine 5 carboxylic acid 6 chloroisoquinolin 1 amine 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 amine 4 4 dimethylimidazolidin 2 one 2 2 difluoro 1 pyridin 2 yl ethanone 3 fluoropicolinaldehyde 1H imidazo 4 5 b pyridin 2 amine 2 chloro 6 trifluoromethyl nicotinonitrile 4 bromobenzofuran 2 carboxylic acid 2 chloro 5 formylphenylboronic acid 2 1H pyrazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 3 amino 9 ethylcabazole 4 bromobenzo b thiophene 2 carboxylic acid

3 Chloro 2 methylbenzenesulfonyl chloride 5 Bromo 2 trifluoromethyl benzonitrile 2 Bromo 4 iodoaniline 4 Bromo 3 trifluoromethyl benzaldehyde 2 Bromomethyl 6 methylpyridine 1 Bromo 2 6 difluoro 4 iodobenzene 4 Chloro 3 fluorophenol 2 Ethoxyphenyl isothiocyanate 3 Bromo 2 methylbenzoic acid 2 Fluoro 5 trifluoromethyl benzonitrile 3 Trifluoromethyl benzyl amine 2 AMINO 3 BROMOBENZONITRILE 2 3 5 6 tetrafluorobenzene 1 4 dicarboxylic acid 5 5‘ Bis 2H tetrazole diammonium salt 6 Bromoisoquinoline 2 4 Dibromo 3 nitropyridine 3 Chloro 2 hydroxybenzaldehyde 3 Cyano 4 isopropoxybenzoic acid 2 Amino 6 nitrobenzimidazole 2 5 Dimethoxybenzaldehyde 2 5 Dibromo 3 picoline 4 methoxy 2 6 dimethyl aniline 3 3 difluorocyclobutoxy methyl benzene 2 chloro 5 fluoropyridine 3 carboxylic acid 2 4 trifluoromethyl phenyl piperazine 3 4 methyl 1H imidazol 1 yl 5 trifluoromethyl aniline 4 Difluoro cyclohexylidene acetic acid 2R 3R 4R 5R 2 4 chlorobenzoyloxy methyl 4 fluoro 5 hydroxy 4 methyloxolan 3 yl 4 chlorobenzoate 3R 3 fluoropiperidine hydrochloride 4 fluoro 1H indazol 5 amine

5 bromo 1 methyl 1H pyrazole 3 carboxylic acid 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrazolo 1 5 a pyrimidine 4 amino 2 4 4 dimethyl 2 oxoimidazolidin 1 yl N 3 trifluoromethyl phenyl pyrimidine 5 carboxamide 2 phenyloxazolo 5 4 b pyridine 7H spiro furo 3 4 b pyridine 5 4 piperidin 7 one 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 hydroxyisonicotinaldehyde 6 bromo 3 methyl 2 trifluoromethyl pyridine 3 5 bis trifluoromethyl phenyl octanamide 7 bromobenzo b thiophene 2 carboxylic acid 4 chlorobenzofuran 2 carboxylic acid 2 borono 4 fluorobenzoic acid 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl piperidin 4 one 2 Chloro 6 fluorophenyl methanesulfonyl chloride 2 Bromo 5 trifluoromethyl benzonitrile 5 Bromo 2 3 6 trifluorobenzaldehyde 2 Bromo 5 methyl 3 nitropyridine 2 Acetylnaphthalene 4 Bromo 2 fluoro 5 trifluoromethyl aniline 1 Bromo 3 5 difluorobenzene 4 Chloro 2 fluorophenol 2 Trifluoromethyl benzyl amine 3 5 Dimethylphenyl isothiocyanate 2 Fluoro 4 trifluoromethyl benzonitrile 2 Bromo 5 methylbenzoic acid 2 BROMO 3 4 DIFLUOROANILINE 2 3 5 6 Tetrafluorobenzyl alcohol 3 5 Dichloro 2 Bromopyridine 4 2 Aminoethyl 1 Boc piperidine 3 Trifluoromethylphenol

5 Amino 6 methylbenzimidazolone 4 Bromo 2 nitroaniline 5 Bromo 2 fluoro 3 picoline 4 Hydroxymethyl piperidine 1 sulfonyl fluoride 4 IODOPYRIDIN 2 AMINE 2 3 4 fluorophenyl oxetan 3 yl ethan 1 ol 5 fluoropyridine 3 carboxylic acid 2R 3R 2 2 4 difluorophenyl 1 1H 1 2 4 triazol 1 yl butane 2 3 diol methanesulfonic acid 1 tert butoxy carbonyl amino 3 3 difluorocyclopentane 1 carboxylic acid 6 fluoro 1H 1 3 benzodiazole 2 carboxylic acid 4 4 Difluoro cyclohexylidene acetic acid 2R 3R 4R 5R 5 bromo 3 4 chlorobenzoyloxy 4 fluoro 4 methyloxolan 2 yl methyl 4 chlorobenzoate 3 fluoro 2 trifluoromethyl pyridine 3S 3 fluoropiperidine hydrochloride 2 chloro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 1H imidazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 6 chloro 3 methyl 2 trifluoromethyl pyridine 3 fluoro 4 iodopyridine 2 chlorooxazolo 5 4 b pyridine 7H Spiro furo 3 4 b pyridine 5 4 piperidin 7 one hydrochloride 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 7 3 chloropropoxy 4 hydroxy 6 methoxyquinoline 3 carbonitrile 4 6 dichlorobenzofuran 6 7 dihydro 5H pyrrolo 3 4 b pyrazine 6 bromopyrazolo 1 5 a pyrimidine 7 methylbenzo b thiophene 2 carboxylic acid 5 acetyl 2 chlorophenylboronic acid 2 Bromo 4 trifluoromethyl benzonitrile 2 Chloro 4 nitrobenzenesulfonyl chloride 4 Fluoro 1 3 benzoxazol 2 3H one