4 4 1E 1 E 2 2 1 phenyl 1H pyrazole 3 5 diyl bis ethene 2 1 diyl bis 2 methoxyphenol 1 8 diazaspiro 5 5 undecan 7 one 1 benzhydryl 3 3 difluoroazetidine 1 benzhydrylamino 3 chloropropan 2 ol 2 2 4 dimethylphenyl phthalazin 1 2H one 1 2 4 dimethylphenyl 2 3 methoxyphenyl diazene 2 OXA SPIRO 3 3 HEPTAN 6 ONE 2 methylpiperidine 2 carboxylic acid hydrochloride 1 Propanone 1 2 4 difluorophenyl 2 hydroxy 2R 1 oxa 3 9 diazaspiro 5 5 undecan 2 one hydrochloride 8 methoxycarbonyl octanoic acid 2R 4S 1 tert Butoxycarbonyl 4 fluoropyrrolidine 2 carboxylic acid 3 fluorotetrahydro 2H pyran 4 yl methanesulfonate 2 1 ADAMANTANYL ETHYL ACETATE 4 methylsulfonyl 2 trifluoromethyl benzaldehyde 4 2 Oxo 2 2 oxo 4 R phenyl oxazolidin 3 yl ethyl piperidine 1 carboxylic acid tert butyl ester 1 bromomethyl 2 trifluoromethyl 4 methylsulfonyl benzene 5 hydroxy 5 trifluoromethyl dihydrofuran 2 3H one 4 4 difluoro N S 3 1S 3R 5R 2 fluoro 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl adamantanecarboxamide 3 3 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl piperidine 4 carboxamide 5 Cyclopropyl 1H pyrazol 3 amine hydrochloride 1 6 Trifluoromethyl pyridin 3 yl ethanone 4 Bromo 2 5 difluorobenzoic acid 2 Trifluoromethyl pyrimidine 4 carboxylic acid 4 Bromo 7 methoxy 1H indole 1 Methylcyclopropanamine hydrochloride 3 5 Difluoro 4 nitrobenzonitrile 3 5 Dibromo 4 methoxypyridine 2 4 Bromo 3 fluorophenyl acetonitrile 4 5 6 7 Tetrahydro 1H benzo d imidazole 5 carboxylic acid hydrochloride

2 Benzo d 1 3 dioxol 5 yl 2 oxoacetaldehyde hydrate 1 3 dibromo 2 chlorobenzene 3 5 Dichloro 2 iodopyrazine 1 Pyridin 3 yl piperazine hydrochloride 2 Oxopiperidine 4 carboxylic acid 6 Bromo 2 phenyl 1H imidazo 4 5 b pyridine 3 Iodo 4 nitrophenol 4 5 Bromo 1 3 4 thiadiazol 2 yl morpholine 4 Amino 6 bromo 2 methylpyrimidine 4 Ethyl 1H pyrazol 3 amine oxalate 3 Dimethylamino phenyl boronic acid hydrochloride 3 Bromo 1 methyl 1H pyrazol 5 amine 7 methoxynaphthalen 1 ol 2 Methoxy 6 trifluoromethyl aniline 4 Piperazin 1 yl pyrimidine 3 Methylimidazo 2 1 b thiazole 2 carboxylic acid 6 Bromo 3 iodopyrazolo 1 5 a pyrimidine 1 Benzylpiperidin 3 amine hydrochloride 1 Isoquinolin 1 ylmethanamine 2 Chloro 7 trifluoromethylquinoxaline 2 Iodo 1 3 dimethoxybenzene 4 Methylthiophene 3 carboxylic acid 1 3 Dimesitylimidazolidin 2 ylidene 2 isopropoxybenzylidene ruthenium VI chloride 5 Amino 2 ethyl 2H indazole 7 Bromo 4 chloro 3 nitroquinoline 2 Hydroxy 4 methoxybenzonitrile 2 Bromo 4 methylpentanoic acid 3 Chloroquinoxaline 2 carboxylic acid 1 Ethylpiperidin 4 yl methanol 1 Thiophen 2 yl piperazine

3 4 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl propanamide 4 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 propanenitrile 3 Fluoro 5 methoxy phenol 3 Amino 1H indazole 5 carbonitrile 2 Amino 3 methoxy 4 fluorobenzoic acid 2 Chloro 3 2 methoxyethyl amino naphthalene 1 4 dione 1H Pyrrolo 2 3 b pyridin 6 ol 4 Methylquinolin 7 amine 2 Amino 2 pyridin 3 yl ethanol 6 Bromoisoquinolin 3 ol 4 Bromo 3 Chloro Benzonitrile 1 Bromomethyl 4 fluoro 2 methoxybenzene 1 Boc 3 bromo 7 nitroindole 1 Bromo 2 iodo 4 trifluoromethyl benzene 6 Chloro 1 2 3 4 tetrahydroquinoline 4 Chloro 2 hydroxybenzonitrile 3 4 Bromophenyl 1H 1 2 4 triazole 1 Methyl 1H 1 2 4 triazol 3 yl methanol 1 Methyl 1H 1 2 4 triazole 3 carboxylic acid methyl ester 1 6 Dioxaspiro 2 5 octane 3 5 Dibromo 2 chloropyrazine 3 6 Dichloropyridazine 4 carbonitrile 4 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 acetamide 4 Bromo N methylpyrimidin 2 amine 3 Oxabicyclo 3 1 0 hexane 6 carboxylic acid 4 Chloro 3 5 difluorobenzonitrile 6 Trifluoromethyl pyridazin 3 2H one 4 1 3 Thiazol 2 yl phenyl methylamine 2 4 Dichloro 5 cyanothiazole 5 2 Methoxyethoxy pyrazin 2 amine

5 2 5 Dichlorophenyl 1H pyrazole 3 carboxylic acid 1 Chloroisoquinoline 4 carbonitrile 6 Methoxy 1 2 3 4 tetrahydropyrido 2 3 b pyrazine 3 4 Dimethylbenzyl bromide 2 Methoxy 6 methylbenzonitrile 3 Bromo 2 Chlorobenzoic acid 4 Bromo 6 hydroxypyrimidine 4 Bromopyrimidin 2 yl cyclohexylamine 1 Methyl 1H imidazo 4 5 b pyridine 2 Amino 5 bromo 6 methylpyrazine 1 2 Diamino 3 chlorobenzene 5 4 Fluorophenethylsulfonyl 1 phenyl 1H tetrazole 2 Chloro 4 methylpyrimidin 5 amine 2 4 Dichloro 6 nitropyridine 1 Methyl 3 azetidinecarboxylic acid 5 Trimethylsilyl ethynyl pyrimidine 2 Chloro 7 methylquinoxaline 4 methyl 2 nitro 1 trifluoromethyl benzene 4 Bromobenzo d isoxazol 3 amine 3 4 Methylpiperazin 1 yl phenyl methanol 1 4 5 6 Tetrahydrocyclopenta c pyrazole 3 carbohydrazide 1 Cyclopentylmethyl piperazine 4 Nitro 2 trifluoromethyl benzenol 2 Bromo N hexadecylacetamide 6 Bromo 2 chloro 3 iodopyridine 3 Iodo 1H pyrazole 2 Bromo 5 nitrobenzenecarbaldehyde 4 Bromo 2 chloro 5 methylpyridine 4 Hydroxytetrahydro 2H thiopyran 1 1 dioxide 5 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl isoindolin 1 one