3 Fluoro 4 methylcarbamoyl phenylboronic acid 2 5 Difluoro 4 formylphenylphenylboronic acid 5 Tert butylcarbmoyl 2 fluorophenylboronic acid 4 Bromo 2 hydroxyphenylboronic acid 3 Morpholinomethyl phenylboronic acid 3 Fluoro 4 morpholinylmethyl phenylboronic acid 1 Tetrahydro pyran 2 yl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 2 Fluoro 6 iodophenylboronic acid pinacol ester 4 4 Methylpiperazino methylphenylboronic acid pinacol ester 2 Chloro 5 methoxymethylphenylboronic acid pinacol ester 2 Fluoro 5 pyrolidine 1 carbonyl phenylboronic acid 2 Fluoro 5 propylcarbamoyl phenylboronic acid 5 Dimethylcarbamoyl 2 fluorobenzeneboronic acid 5 Carbamoyl 2 fluorophenyboronic acid 2 5 Difluoro 4 benzyloxyphenylboronic acid 2 Fluoro 5 methoxypyridine 3 boronic acid 4 4 5 5 Tetramethyl 2 3 trifluoromethyl benzyl 1 3 2 dioxaborolane 4 Methoxymethyl 2 6 dimethylphenylboronic acid 6 Bromo 2 methylpyridine 3 boronic acid pinacol ester 4 Bromo 2 5 bifluorophenylboronic acid 2 5 Difluoro 4 methoxymethoxy phenylboronic acid 2 3 Difluoro 4 hydroxyphenylboronic acid pinacol ester 4 Methoxycarbonyl 3 5 difluorophenylboronic acid pinacol ester 3 5 Difluoro 2 methylsulfanylphenylboronic acid 3 Chloro 2 cyanophenylboronic acid 3 Bromo 2 6 dichlorophenylboronic acid 2 Bromo 4 fluorophenylboronic acid 4 Bromo 3 carboxyphenylboronic acid 4 1 3 Dioxolan 2 yl 2 6 difluorophenylboronic acid 3 4 Difluoro 2 isopropoxyphenylboronic acid

4 Phenylamino methyl phenylboronic acid 3 4 Difluoro 2 ethoxyphenylboronic acid 5 Benzyloxy 2 methylphenylboronic acid 4 Bromo 3 methylphenylboronic acid N butyldiethanolamine ester 4 Benzyloxy 2 trifluoromethyl phenylboronic acid 4 Butoxy 3 5 dichlorophenylboronic acid 3 5 Dichloro 4 isopropoxyphenyboronic acid 2 Methoxy 5 methylaminocarbonyl phenylboronic acid 2 Acetylphenylboronic acid pinacol ester 4 Bromo 3 ethoxycarbonyl 2 fuorophenylboronic acid 2 6 Dichloro 3 formylphenylboronic acid 3 5 Dichloro 4 formylphenylboronic acid 4 Bromo 2 3 dimethylphenylboronic acid 3 5 Difluoro 4 iodophenylboronic acid 4 Hydroxymethyl 2 methoxyphenylboronic acid 6 Bromo 2 3 dichlorophenylboronic acid 2 Methyl 5 cyanophenylboronic acid pinacol ester 3 Bromo 5 fluorophenylboronic acid N butyldiethanolamine ester 2 4 Difluoro 3 methoxycarbonylphenylboronic acid 5 Amino 2 fluorobenzeneboronic acid pinacol ester 2 Methylthiophene 3 boronic acid pinacol ester 2 Chloro 5 isopropylphenyl boronic acid 5 Bromo 2 isopropoxy pyridine 4 boronic acid 4 Methoxymethoxy 2 6 dimethylphenylboronic acid 4 N N Diethylaminocarbonyl phenylboronic acid pinacol ester 2 6 Difluoro 3 isopropoxyphenylboronic acid 2 Fluoro 3 N N dimethylaminocarbonyl phenylboronic acid 4 Chloro 3 fluoro 2 formylphenylboronic acid 4 Methoxycarbonyl 3 trifluoromethyl phenylboronic acid 2 Fluoro 3 carboxypyridine 5 boronic acid

3 5 Dimethy 4 hydroxyphenylboronic acid pinacol ester 4 Chloro 3 5 difluorophenylboronic acid pinacol ester 3 5 Dimethylbiphenyl 4 ylboronic acid 2 6 Dimethyl 4 ethoxyphenylboronic acid 2 5 Dibromo 4 pyridinylboronic acid pinacol ester 3 Bromo 2 isopropoxy 5 formylphenylboronic acid 2 tert Butylcarbonylamino 6 chlorophenylboronic acid 5 Bromo 3 methylpyridine 4 boronic acid 5 Carboxypyridine 3 boronic acid 3 Diethylcarbamoyl 2 fluorophenylboronic acid 3 5 Bis trifluoromethyl 2 bromophenylboronic acid 5 Formyl 2 methylphenylboronic acid 2 4 Di tert butoxy pyrimidine 5 carboxaldehyde 4 Acetyl 2 3 difluorophenylboronic acid 2 Pyrrolidin 1 ylpyrimidin 5 yl boronic acid 2 Ethoxy 3 methylpyridine 5 boronic acid 4 Formyl 2 trifluoromethyl phenylboronic acid 5 Bromo 2 trifluoromethoxyphenylboronic acid 2 Chloro 6 methoxypyridine 3 lboronic acid 4 Fluorophenylboronic acid N butyldiethanolamine ester 2 Fluoro 5 methylpyridine 4 boronic acid 4 Aminocarbonyl 3 5 difluorophenylboronic acid 4 Chloro 3 trifluoromethoxy phenylboronic acid 3 Formyl 5 trifluoromethoxy phenylboronic acid pinacol ester 2 Fluoro 4 piperidine 1 carbonyl phenylboronic acid 2 Fluoro 4 N ethylaminocarbonyl phenylboronic acid 4 N Methylaminocarbonyl 2 fluorophenylboronic acid 3 Formyl 5 trifluoromethoxy phenylboronic acid 3 Benzyloxyphenylboronic acid pinacol ester 4 1 1 dimethylethoxy carbonyl phenylmethyl aminophenylboronic acid

3 Hydroxymethyl 4 trifluoromethoxy phenylboronic acid 5 Formyl 3 methoxyphenylboronic acid 5 Hydroxymethyl 2 methoxyphenylboronic acid 3 5 Dimethyl 4 hydroxyphenylboronic acid 2 Methoxymethoxy 5 trifluoromethyl phenylboronic acid 3 Fluoro 5 morpholine 4 carbonyl phenylboronic acid 4 Ethoxy 3 5 dichlorophenylboronic acid 5 Dimethylcarbamoyl 3 fluorophenylboronic acid 3 Aminocarbonyl 5 fluorophenylboronic acid 3 Fluoro 5 diethylcarbamoyl phenylboronic acid 4 Methylthio 2 trifluoromethyl phenylboronic acid 3 Fluoro 5 methylcarbamoyl phenylboronic acid 5 Fluoro 3 formyl 2 methoxyphenylboronic acid 3 Bromo 5 methoxycarbonyl phenylboronic acid 2 3 Dichloro 6 trifluoromethyl benzoic acid 3 Ethoxy 5 fluorophenylboronic acid 4 Chloro 2 fluoro 3 hydroxyphenylboronic acid 3 Piperidin 1 ylmethyl phenylboronic acid 4 Bromo 2 chlorophenylboronic acid 4 Bromo 2 ethylphenylboronic acid 4 Carboxy 3 trifluoromethyl phenylboronic acid 4 Benzyloxy 2 3 difluorophenylboronic acid 2 Fluoro 6 phenoxyphenylboronic acid 3 Fluoro 2 formyl 6 methoxyphenylboronic acid 4 Bromo 3 formylphenylboronic acid 2 Bromo 6 fluoro 3 hydroxyphenylboronic acid 2 Bromo 3 iodophenylboronic acid 5 Carboxy 4 chloro 2 fluorophenylboronic acid 2 3 Dimethoxy 6 fluorophenylboronic acid 5 Hydroxymethyl 2 methylphenylboronic acid