3 4 Ethylenedioxybenzene boronic acid pinacol ester 2 Phenylethyl 1 boronic acid pinacol ester 2 6 Dimethyl 4 chlorophenylboronic acid 4 Amino 2 methylphenylboronic acid pinacol ester 4 2 Morpholinoethoxy phenylboronic acid pinacol 6 Bromo 2 fluoro 3 propoxyphenylboronic acid 4 Carboxy 3 methylphenylboronic acid 4 Methyl 3 nitrophenylboronic acid pinacol ester 4 4 Bromophenylcarbamoyl phenylboronic acid 4 2 Carbamothioylhydrazinecarbonyl phenylboronic acid 2 Fluoro 4 methylthiophenylboronic acid 4 Benzyloxy 3 methoxyphenylboronic acid 3 2 4 Dimethylphenylcarbamoyl phenylboronic acid 4 Benzyloxycarbonylphenylboronic acid pinacol ester 2 Methoxy 5 methoxycarbonylphenylboronic acid pinacol ester 1 Propyl 1H pyrazole 5 boronic acid pinacol ester 2 Amino 5 fluorophenyl boronic acid pinacol ester 3 Fluoro 4 methoxymethoxy phenylboronic acid 2 Methoxymethoxy 5 methylphenylboronic acid 3 Methoxymethoxy 4 methylphenylboronic acid 4 Fluoro 3 pyrrolidine 1 carbonyl phenylboronic acid 4 Fluoro 3 piperidine 1 carbonyl phenylboronic acid 3 Fluoro 4 hydrazinocarbonylphenylboronic acid 3 Carboxy 5 nitrophenylboronic acid pinacol ester 5 Chloro 2 isopropoxyphenylboronic acid 3 Amino 4 chlorophenylboronic acid pinacol ester 4 Chloro 3 methylphenylboronic acid 2 Chloro 6 fluoro 3 methylphenylboronic acid 2 Chloro 6 fluorophenylboronic acid 2 Cyanophenylboronic acid neopentyl ester

4 Cyclopentylphenylboronic acid 3 Chlorophenylboronic acid pinacol ester 2 Carboxy 5 pyridineboronic acid 6 Phenylpyridine 3 boronic acid 2 6 Dibromo 3 methoxyphenylboronic acid 3 5 Dinitro 2 methylphenylboronic acid 2 4 Difluorophenylboronic acid pinacol ester 3 Ethoxycarbonyl 5 nitrophenylboronic acid 2 Fluoro 3 iodophenylboronic acid 5 Fluoro 2 formylphenylboronic acid 3 Formylphenylboronic acid pinacol ester 4 Fluoro 2 propoxyphenylboronic acid 4 Hydroxymethyl 2 6 difluorophenylboronic acid 4 Hydroxy 2 trifluoromethyl phenylboronic acid 4 4 Isopropoxyphenyl phenylboronic acid 2 Isopropoxy 4 trifluoromethyl phenylboronic acid 4 Isobutylphenylboronic aicd pinacol ester 2 Methylthio phenylboronic acid pinacolate 2 Methoxycarbonyl 3 fluorophenylboronic acid 4 Methoxy 3 nitrophenylboronic acid 2 Methoxyphenylboronic acid pinacol ester 4 Methoxymethylphenylboronic acid 3 Nitrophenylboronic acid pinacol ester 3 Bromo 5 methylphenylboronic acid 2 Bromo 6 fluorophenylboronic acid 2 Butoxy 5 fluorophenylboronic acid 3 Butoxycarbonylphenylboronic acid 3 Bromomethyl benzeneboronic acid neopentyl glycol ester 3 Bromo 5 methyl 2 methoxyphenylboronic acid 3 Bromo 2 isopropoxy 5 methylphenylboronic acid

4 Butoxy 3 fluorophenylboronic acid 2 Benzyloxy 3 bromo 5 methylphenylboronic acid 3 Amino 4 methylphenylboronic acid hydrochloride 5 Acetyl 2 methoxyphenylboronic acid 3 Amino 4 chlorophenylboronic acid 4 Ethoxycarbonyl 3 methoxyphenylboronic acid 3 Formyl 4 methylphenylboronic acid 2 5 Dichloropyridine 4 boronic acid pinacol ester 4 tert Butyl dimethylsiloxy phenyl boronic acid 4 Formyl 3 methylphenylboronic acid 5 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 carboxylic acid diethylamide 3 Chloro 2 methylphenyboronic acid 5 Bromo 2 methoxypyridine 3 boronic acid 2 5 Dibromopyridine 3 boronic acid pinacol ester 4 Benzyloxy 2 piperidine 1 yl pyrimidine 5 boronic acid 5 Chloro 2 trifluoromethyl phenylboronic acid 4 Benzyloxy 2 piperidine 1 yl pyrimidine 5 boronic acid pinacol ester 3 Bromo 2 6 difluorophenylboronic acid 2 Cyano 3 5 5 Dimethyl 1 3 2 dioxaborinan 2 yl pyridine 3 Chloro 5 trifluoromethyl phenylboronic acid 2 Chloro 5 hydroxymethylphenylboronic acid 2 Ethoxy 5 fluorophenylboronic acid 2 Bromo 3 methylpyridine 5 boronic acid pinacol ester 6 Methylcarbamoyl pyridin 3 yl boronic acid 1 benzyl 3 3 difluoropiperidin 4 amine 2 3 DIFLUORO 5 NITROPHENOL 4 trifluoromethyl piperidin 4 ol hydrochloride 2 2 2 trifluoro 1 piperidin 4 yl ethanone oxalate 1 1 piperidine 1 3 diyl bis 2 2 2 trifluoroethanone 1 BOC 3 TRIFLUOROMETHYL PIPERIDIN 4 ONE

1 1 benzylpiperidin 3 yl 2 2 2 trifluoroethanone 1 tert butyl 3 methyl 5 5 difluoropiperidine 1 3 dicarboxylate 5 5 difluoropiperidine 3 carboxylic acid hydrochloride 2 4 fluorophenyl 7 8 dimethoxyquinolin 4 1H one 1 tert butoxycarbonyl 5 fluoropiperidine 3 carboxylic acid 3 fluoromethylpiperidine HCl salt 1 benzyl 3 3 difluoropiperidin 4 ol 1 piperidin 4 yl 1H indole trifluoroacetate 1 benzyl 3 2 2 2 trifluoroacetyl piperidin 4 one hydrochloride 2 2 2 trifluoro 1 4 4 methylbenzoyl piperidin 1 yl ethanone 1 BENZYL 1 2 DIHYDRO 5 FLUORO 2 OXO SPIRO 3H INDOLE 3 4 PIPERIDINE 2 1 tert butoxycarbonyl piperidin 4 yl 2 2 difluoroacetic acid 3 3 difluorocyclopentanecarboxylic acid 75 solution in EtOAc and CH2Cl2 1 tert butoxycarbonyl 3 fluoropiperidine 4 carboxylic acid 1 1 9H fluoren 9 yl methoxy carbonyl pyrrolidin 3 yl piperidine 3 carboxylic acid 1 tert butyl 3 ethyl 5 5 difluoropiperidine 1 3 dicarboxylate 1 tert butyl 4 ethyl 3 3 difluoro 4 methylpiperidine 1 4 dicarboxylate 3 3 difluoropiperidin 4 ol hydrochloride 1 benzyl 3 methyl 5 5 difluoropiperidine 1 3 dicarboxylate 1 benzyl 4 fluoropiperidin 3 yl methanol 1 tert butyl 3 methyl 4 trifluoromethyl 5 6 dihydropyridine 1 3 4H dicarboxylate 2 1 tert butoxycarbonyl 3 3 difluoropiperidin 4 yl acetic acid 4 benzyl methyl amino 3 5 difluorobenzoic acid 8 Boc 2 fluoro 8 aza bicyclo 3 2 1 octan 3 ol 3 trifluoromethyl piperidin 3 ol hydrochloride 6 fluoro 3 piperidin 4 yl 1H indazole hydrochloride 1 N Boc 4 fluoropiperidine 9 4 bromobutyl 9H fluorene 9 carboxylic acid 4 dimethylamino 3 5 difluorobenzoic acid 2 2 2 trifluoro 1 piperazin 1 yl ethanone hydrochloride