2 Phenylethyl 1 boronic acid pinacol ester 2 6 Dimethyl 4 chlorophenylboronic acid 3 Fluoro 4 hydrazinocarbonylphenylboronic acid 2 Methoxycarbonyl 3 fluorophenylboronic acid 4 Methoxy 3 nitrophenylboronic acid 2 Methoxyphenylboronic acid pinacol ester 4 Methoxymethylphenylboronic acid 3 Nitrophenylboronic acid pinacol ester 2 Methylthio phenylboronic acid pinacolate 4 4 Isopropoxyphenyl phenylboronic acid 2 Isopropoxy 4 trifluoromethyl phenylboronic acid 4 Isobutylphenylboronic aicd pinacol ester 4 Fluoro 2 propoxyphenylboronic acid 4 Hydroxymethyl 2 6 difluorophenylboronic acid 4 Hydroxy 2 trifluoromethyl phenylboronic acid 3 Formylphenylboronic acid pinacol ester 5 Fluoro 2 formylphenylboronic acid 3 Ethoxycarbonyl 5 nitrophenylboronic acid 3 5 Dinitro 2 methylphenylboronic acid 2 4 Difluorophenylboronic acid pinacol ester 2 Fluoro 3 iodophenylboronic acid 2 6 Dibromo 3 methoxyphenylboronic acid 6 Phenylpyridine 3 boronic acid 2 Carboxy 5 pyridineboronic acid 3 Chlorophenylboronic acid pinacol ester 2 Chloro 6 fluorophenylboronic acid 2 Cyanophenylboronic acid neopentyl ester 4 Cyclopentylphenylboronic acid 3 Amino 4 chlorophenylboronic acid pinacol ester 2 Chloro 6 fluoro 3 methylphenylboronic acid

4 Chloro 3 methylphenylboronic acid 5 Chloro 2 isopropoxyphenylboronic acid 3 Bromo 2 isopropoxy 5 methylphenylboronic acid 4 Butoxy 3 fluorophenylboronic acid 3 Carboxy 5 nitrophenylboronic acid pinacol ester 3 Bromo 5 methyl 2 methoxyphenylboronic acid 2 Butoxy 5 fluorophenylboronic acid 3 Butoxycarbonylphenylboronic acid 3 Bromomethyl benzeneboronic acid neopentyl glycol ester 3 Amino 4 methylphenylboronic acid hydrochloride 5 Acetyl 2 methoxyphenylboronic acid 2 Benzyloxy 3 bromo 5 methylphenylboronic acid 3 Bromo 5 methylphenylboronic acid 2 Bromo 6 fluorophenylboronic acid 3 Formyl 4 methylphenylboronic acid 5 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 carboxylic acid diethylamide 4 Formyl 3 methylphenylboronic acid 2 5 Dichloropyridine 4 boronic acid pinacol ester 3 Amino 4 chlorophenylboronic acid 4 Ethoxycarbonyl 3 methoxyphenylboronic acid 5 Bromo 2 methoxypyridine 3 boronic acid 4 tert Butyl dimethylsiloxy phenyl boronic acid 3 Chloro 2 methylphenyboronic acid 2 Chloro 5 hydroxymethylphenylboronic acid 2 Ethoxy 5 fluorophenylboronic acid 2 Bromo 3 methylpyridine 5 boronic acid pinacol ester 2 5 Dibromopyridine 3 boronic acid pinacol ester 4 Benzyloxy 2 piperidine 1 yl pyrimidine 5 boronic acid 5 Chloro 2 trifluoromethyl phenylboronic acid 4 Benzyloxy 2 piperidine 1 yl pyrimidine 5 boronic acid pinacol ester

3 Bromo 2 6 difluorophenylboronic acid 3 Chloro 5 trifluoromethyl phenylboronic acid 2 Cyano 3 5 5 Dimethyl 1 3 2 dioxaborinan 2 yl pyridine 6 Methylcarbamoyl pyridin 3 yl boronic acid 1 benzyl 3 3 difluoropiperidin 4 amine 2 3 DIFLUORO 5 NITROPHENOL 1 1 piperidine 1 3 diyl bis 2 2 2 trifluoroethanone 1 BOC 3 TRIFLUOROMETHYL PIPERIDIN 4 ONE 1 benzyl 3 2 2 2 trifluoroacetyl piperidin 4 one hydrochloride 2 2 2 trifluoro 1 4 4 methylbenzoyl piperidin 1 yl ethanone 4 trifluoromethyl piperidin 4 ol hydrochloride 2 2 2 trifluoro 1 piperidin 4 yl ethanone oxalate 1 1 benzylpiperidin 3 yl 2 2 2 trifluoroethanone 1 piperidin 4 yl 1H indole trifluoroacetate 3 fluoromethylpiperidine HCl salt 1 benzyl 3 3 difluoropiperidin 4 ol 1 BENZYL 1 2 DIHYDRO 5 FLUORO 2 OXO SPIRO 3H INDOLE 3 4 PIPERIDINE 1 tert butyl 3 methyl 5 5 difluoropiperidine 1 3 dicarboxylate 5 5 difluoropiperidine 3 carboxylic acid hydrochloride 2 4 fluorophenyl 7 8 dimethoxyquinolin 4 1H one 1 tert butoxycarbonyl 5 fluoropiperidine 3 carboxylic acid 3 3 difluorocyclopentanecarboxylic acid 75 solution in EtOAc and CH2Cl2 2 1 tert butoxycarbonyl piperidin 4 yl 2 2 difluoroacetic acid 1 tert butoxycarbonyl 3 fluoropiperidine 4 carboxylic acid 1 1 9H fluoren 9 yl methoxy carbonyl pyrrolidin 3 yl piperidine 3 carboxylic acid 1 tert butyl 4 ethyl 3 3 difluoro 4 methylpiperidine 1 4 dicarboxylate 1 benzyl 3 methyl 5 5 difluoropiperidine 1 3 dicarboxylate 3 3 difluoropiperidin 4 ol hydrochloride 1 benzyl 4 fluoropiperidin 3 yl methanol 1 tert butyl 3 ethyl 5 5 difluoropiperidine 1 3 dicarboxylate

1 tert butyl 3 methyl 4 trifluoromethyl 5 6 dihydropyridine 1 3 4H dicarboxylate 2 1 tert butoxycarbonyl 3 3 difluoropiperidin 4 yl acetic acid 4 benzyl methyl amino 3 5 difluorobenzoic acid 8 Boc 2 fluoro 8 aza bicyclo 3 2 1 octan 3 ol 3 trifluoromethyl piperidin 3 ol hydrochloride 1 N Boc 4 fluoropiperidine 6 fluoro 3 piperidin 4 yl 1H indazole hydrochloride 4 dimethylamino 3 5 difluorobenzoic acid 2 2 2 trifluoro 1 piperazin 1 yl ethanone hydrochloride 4 chloro 3 fluoropyridine 1 benzyl 3 trifluoromethyl piperidin 4 ol 2 2 difluoropentanedioic acid 1 benzyl 3 trifluoromethyl piperidin 4 one 3 trifluoromethyl pyrrolidine hydrochloride 2 TRIFLUOROMETHOXY ETHYLAMINE HYDROCHLORIDE 1 benzyl 3 fluoro 1 2 5 6 tetrahydropyridin 4 yl methanol 3 4 Cis 1 tert butyl 4 methyl 3 fluoropiperidine 1 4 dicarboxylate racemate 1 amino 3 fluoropropan 2 ol hydrochloride 3 3 difluoro 1 4 bipiperidine dihydrochloride 4 fluoro 1 hydroxymethyl admantane 4 4 difluoro 1 hydroxymethyladmantane 1 N Boc 4 4 difluoropiperidine 3 3 difluoro 4 4 fluorobenzyl piperidine hydrochloride 5 5 difluoropiperidin 3 yl methanol hydrochloride 3 Iodo 2 phenoxypyridine 7 7 difluoro 4 5 6 7 tetrahydro 1H pyrazolo 4 3 c pyridine hydrochloride 3 acetamido 6 acetyl 2 nitrophenyl 4 benzyl methyl amino 3 5 difluorobenzoate 3 acetamido 2 nitrophenyl 4 benzyl methyl amino 3 5 difluorobenzoate 3 acetamido 2 nitrophenyl 4 dimethylamino 3 5 difluorobenzoate 3S 4R 1 tert butoxycarbonyl 3 fluoropiperidine 4 carboxylic acid enantiomer b 87 e e