4 Hydroxymethyl 3 methylphenylboronic acid 2 3 Dimethyl 4 formylphenylboronic acid 4 Formyl 3 isopropylphenylboronic acid 2 Formyl 5 trifluoromethoxy phenylboronic acid 5 Formylpyridine 3 boronic acid 3 6 Difluoro 2 methoxyphenylboronic acid 3 Ethoxy 4 methylphenylboronic acid 3 Isoproproxy 4 methylphenylboronic acid 2 4 Difluoro 6 bromophenylboronic acid 5 Ethoxypyridine 3 boronic acid 3 3 chloro 4 fluorophenylcarbamoyl 4 fluorophenylboronic acid 3 3 5 dichlorophenylcarbamoyl 4 fluorophenylboronic acid 3 4 Bromo 2 6 dimethylphenylcarbamoyl 4 fluorophenylboronic acid 2 Isopropylboronic acid pinacol ester 4 Chloro 3 ethylphenylboronic acid 5 Carboxy 2 ethoxyphenylboronic acid 3 5 Bis trifluoromethyl benzylboronic acid 2 Fluoro 4 formylphenylboronic acid 4 Fluoro 3 N methoxy N methyl carbamoyl phenylboronic acid 4 Fluoro 3 N propylcarbamoyl phenylboronic acid 4 Fluoro 3 morpholine 4 carbonyl phenylboronic acid 4 Fluoro 3 methylcarbamoyl phenylboronic acid 2 Amino 4 methylphenylboronic acid pinacol ester 5 Bromo 2 hydroxyphenylboronic acid 4 Methyl 2 nitrophenylboronic acid pinacol ester 3 2 5 Dimethylphenylcarbamoyl phenylboronic acid 3 2 3 Dimethylphenylcarbamoyl phenylboronic acid 6 Hydroxymethyl pyridine 3 boronic acid 3 3 Fluorophenylcarbamoyl phenylboronic acid 3 2 Bromophenylcarbamoyl phenylboronic acid

4 Diethylcarbamoyl 2 methoxyphenylboronic acid 4 3 Fluorophenylcarbamoyl phenylboronic acid 4 4 Chlorophenylcarbamoyl phenylboronic acid 5 Bromo 2 chloropyridine 3 boronic acid 4 Formyl 3 trifluoromethyl phenylboronic acid 3 Hydroxy 4 methoxyphenylboronic acid pinacol ester 6 Bromo 4 methylpyridine 3 boronic acid 3 Chloro 5 formylphenylboronic acid 6 4 4 5 5 Tetramethyl1 3 2 dioxaboralan 2 yl 2 3 dihydroinden 1 one 6 Bromo 2 fluoro 3 iodophenylboronic acid 2 Methyl 4 carboxyphenylboronic acid 5 Carboxy 2 methoxyphenylboronic acid 5 Chloro 2 pivaloylamino phenylboronic acid 2 Benzyloxy 5 formylphenylboronic acid 4 Amino 3 chlorobenzeneboronic acid pinacol ester 4 Amino 2 fluorophenylboronic acid pinacol ester 5 Phenyl 2 thienylboronic acid 2 Methylthiophene 3 boronic acid 2 Methoxy 4 trifluoromethyl phenylboronic acid 4 Methoxycarbonylphenylboronic acid pinacol ester 3 Tetrahydro 2H pyran 2 yloxy phenylboronic acid 5 Hydroxymethylfuran 2 boronic acid 4 Fluoro 2 isopropoxyphenylboronic acid 2 Fluoro 5 isoproproxyphenylboronic acid 2 4 Dichloro 5 nitrophenylboronic acid 3 5 Dichloro 4 methoxyphenylboronic acid 2 Ethoxy 5 methylphenylboronic acid 4 Bromopyridine 3 boronic acid 3 Chloro 2 4 difluorophenylboronic acid 3 Bromo 2 ethoxy 5 methylphenylboronic acid

2 Methoxycarbonylphenylboronic acid pinacol ester 5 Chloro 2 4 difluorophenylboronic acid 3 Formylthiophene 2 boronic acid 4 N Butoxy 2 methylphenylboronic acid 4 Benzyloxy 3 5 dimethylphenylboronic acid 2 Benzyloxy 5 methylphenylboronic acid 4 Bromo 2 5 dimethoxyphenylboronic acid 2 Bromo 4 5 difluorophenylboronic acid 3 Bromo 2 fluorophenylboronic acid 2 Bromo 3 ethoxy 6 fluorophenylboronic acid 3 Benzyloxycarbonyl 5 nitrophenylboronic acid 2 Methoxy 4 methoxycarbonyl phenylboronic acid 2 Bromo 5 6 difluorophenylboronic acid 2 Acetylaminophenylboronic acid pinacol ester 4 Aminocarbonyl phenylboronic acid pinacol ester 5 Formyl 2 ethoxyphenylboronic acid 3 Methylthiophenylboronic acid pinacol ester 4 Ethoxy 2 formylphenylboronic acid 2 4 Dimethoxyphenylboronic acid pinacol ester 2 3 Difluoro 4 n hexyloxy phenylboronic acid 4 Fluorophenylboronic acid pinacol ester 2 Chloro 6 trifluoromethylbenzoic acid 3 Chloro 4 formylphenylboronic acid 1 Hexaneboronic acid cyclic iminodiethylene ester 4 Formyl 2 methylphenylboronic acid 3 Tetrahydro 2H pyran 2 yloxy phenylboronic acid pinacol ester 2 Chloro 6 isopropylpyridine 3 boronic acid 3 Bromo 2 chloropyridine 4 boronic acid pinacol ester 3 FLUOROPIPERIDINE HYDROCHLORIDE 1 1 piperidine 1 4 diyl bis 2 2 2 trifluoroethanone

2 2 2 trifluoro 1 4 4 fluorobenzoyl piperidin 1 yl ethanone 3 difluoromethylpiperidine hydrochloride 3 fluoro adamantane 1 methanol 5 6 chloropyridazin 3 yl methyl 2 2 fluorophenyl 5H imidazo 4 5 c pyridine 3 Cyano 4 5 5 Dimethyl 1 3 2 dioxaborinan 2 yl pyridine 4 Cyano 3 5 5 Dimethyl 1 3 2 dioxaborinan 2 yl pyridine 5 6 2 4 bis trifluoromethyl phenyl pyridazin 3 yl methyl 2 2 fluorophenyl 5H imidazo 4 5 c pyridine 4 4 difluoropiperidin 3 ol hydrochloride 1 tert butoxycarbonyl 5 5 difluoropiperidine 2 carboxylic acid 1 1 benzylpiperidin 4 yl 2 2 2 trifluoroethanone oxalate 1 4 2 4 difluorobenzoyl piperidin 1 yl 2 2 2 trifluoroethanone 4 Hydroxydibenzothiophene 2 3 difluoro 4 nitrophenol 3 3 difluoro 5 hydroxypiperidin 2 one 1 tert butoxycarbonyl 5 5 difluoropiperidine 3 carboxylic acid 1 2 2 2 TRIFLUOROACETYL 4 PIPERIDINECARBOXYLIC ACID 3 amino 2 2 difluoropropanoic acid hydrochloride 4 fluoro 2 methylamino benzoic acid 1 tert butoxycarbonyl 3 3 difluoropiperidine 4 carboxylic acid 3 4 cis 1 benzyloxycarbonyl 3 fluoropiperidine 4 carboxylic acid 1 tert butyl 3 methyl 4 4 difluoropiperidine 1 3 dicarboxylate 1 tert butoxycarbonyl 4 4 difluoropiperidine 3 carboxylic acid 4 4 DIFLUOROADAMANTANE 1 CARBOXYLIC ACID METHYL ESTER 1 benzyl 4 fluoropiperidin 3 yl methyl acetate 1 tert butyl 3 ethyl 5 5 difluoro 4 oxopiperidine 1 3 dicarboxylate 1 benzyl 3 difluoromethylene piperidine 2 1 tert butoxycarbonyl 3 fluoropiperidin 4 yl acetic acid 4 Trifluoroacetyl piperidine hydrochloride 1 tert butyl 4 ethyl 5 fluoro 4 methyl 3 4 dihydropyridine 1 4 2H dicarboxylate 1 tert butyl 3 ethyl 5 fluoropiperidine 1 3 dicarboxylate