2 4 Trifluoromethoxyl phenyl ethanol 3 Methylbenzene 1 2 diamine 5 Fluoro 2 nitrobenzaldehyde 4 Chloro 3 fluoroacetophenone 1 Methylthio 3 trifluoromethyl benzene 5 Bromo 2 iodo 1 3 diethylbenzene 2 5 Dibromopyridine 1 Isopropenyl 4 methoxybenzene 1 3 Bis 2 4 6 trimethylphenyl 4 5 dihydroimidazol 2 ylidene 4 Iodo 4 methylbiphenyl 5 Amino 2 hydroxypyridine 2 Bromo 5 trifluoromethyl pyridine 4 2H benzo d 1 2 3 triazol 2 yl benzene 1 3 diol 4 4 Hydroxy 3 iodophenyl benzonitrile 2 Fluoro 4 iodoaniline 5 fluoropyrazolo 1 5 a pyridine 1 cyclopropyl 6 7 difluoro 1 4 dihydro 4 oxo 1 8 naphthyridine 3 carboxylic acid 1h pyrrolo 3 2 b pyridine 5 carbonitrile 6 fluoro 3 trifluoromethyl 1H indol 6 amine 4 trifluoromethyl 1H pyrrolo 2 3 b pyridine 3 fluoro 4 morpholin 4 yl aniline 1 aminomethyl 4 4 difluorocyclohexan 1 ol 2 3 fluorophenyl pyrrolidine 5 chloro 6 iodoisoindolin 1 one 4 hydroxy N N 2 trimethyl 1 tosyl 1H benzo d imidazole 6 carboxamide 6 methoxy 5 trifluoromethyl pyridin 3 amine 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 3 bromo 2 methoxyphenyl ethanone 2 amino 4 hydroxy 3 methoxybenzoic acid 4 dimethylamino phenyl boronic acid

2 5 chloro 2 fluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 bromo 1H pyrazolo 4 3 b pyrazine 5 fluoro 2 hydroxyphenylboronic acid 5 Methyluracil 6 chloro 3 4 dihydro 2H benzo b 1 4 oxazine 4 Bromo 5 fluoro 2 nitrotoluene 3 Fluorobenzyl bromide 4 Iodobenzoyl chloride 1 2 Difluoro 3 4 5 tribromobenzene 4 Amino 3 trifluoromethyl anisole 2 Bromo 4 cyanoacetophenone 2 Mercapto 6 phenylpyrimidin 4 one 4 Methyl 1 difluoromethoxy benzene 5 Bromo 2 iodo 1 ethylbenzene 4 Methylphenylacetic acid 2 Nitro 4 trifluoromethyl benzoic acid 3 Chlorobenzyl chloride 2 4 Tert butylphenyl ethanol 1 2 Diamino 3 5 difluorobenzene 4 Fluoro 3 nitrobenzaldehyde 3 Chloro 5 fluoroacetophenone 1 Phenyl 1 cyclopropanecarboxylic acid 4 Bromo 9H carbazole 2 Amino 3 Nitro 5 Bromopyridine 5 Bromo 2 hydroxy 3 picoline 4 Bromopiperidine hydrobromide 1 Boc 4 4 Bromobutyl piperidine 3 Chloro 2 fluoroaniline 2 Bromo 3 fluoro 6 methylpyridine 3 Trifluoromethoxy nitrobenzene

3 aMino 6 broMopyrazine 2 carboxylic acid 1 benzyloxy carbonyl 3 fluoroazetidine 3 carboxylic acid 2 amino 5 fluoropyridine 3 carboxylic acid 3 3 4 4 tetrafluoropyrrolidine hydrochloride 1h benzimidazole 2 r 3 methyl 4 2 2 2 trifluoroethoxy 2 pyridinyl methyl sulfinyl 5 fluoro 1H pyrrolo 2 3 b pyridine 3 carbaldehyde 3aS 4R 6aR 6 benzyloxy methyl 5 fluoro 2 2 dimethyl 2H 3aH 4H 6aH cyclopenta d 1 3 dioxol 4 ol 2 2 fluorophenyl pyrrolidine 2 3 dichloro 6 nitroaniline 5 fluoro 2 methoxypyridin 4 amine 3 iodo 1 methyl 1H pyrazole 3 5 dichloropyrazine 2 carboxylic acid 1 5 chloro 2 methoxyphenyl ethanone 2 3 5 bis methoxymethoxy phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 6 fluorobenzo b thiophen 7 yl boronic acid 4 bromo 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 4 hydroxy 3 methylphenylboronic acid 5 nitro 3 4 dihydronaphthalen 1 2H one 3 Bromo 2 fluorotoluene 4 Ethoxybenzyl alcohol 2 3 Difluoroiodobenzene 3 Amino 5 trifluoromethyl anisole 1 Methyl 1H imidazol 2 yl methanol 2 Bromo 3 cyanoacetophenone 4 1H Imidazol 1 yl phenol 2 Hydroxypyrimidine HCl 5 Bromo 2 fluoro 1 ethylbenzene 4 Iodo 1 difluoromethoxy benzene 3 Chloro 4 fluoroacetophenone 4 Fluoro 3 methylbenzaldehyde

4 5 Dichlorobenzene 1 2 diamine 2 Phenylethanol 5 Nitro 2 3 4 trifluorobenzoic acid 2 Methylphenylacetic acid 3 Amino 2 chloropyridine 3 5 Dimethyl 4 2 chloroethyl 1H pyrazole 4 5 Bis diphenylphosphino 9 9 dimethylxanthene 4 Bromo 2 hydroxypyridine 2 Trifluoromethoxy nitrobenzene 5 Amino 2 trifluoromethyl pyridine 4 Bromo 2 fluoroaniline 2 Methylbenzofuro 2 3 b pyridine 8 yl trifluormethanesulfonate 5 bromo 2 trifluoromethyl isonicotinic acid 3aS 4R 6aR 5 fluoro 2 2 dimethyl 6 triphenylmethoxy methyl 2H 3aH 4H 6aH cyclopenta d 1 3 dioxol 4 ol 5 trifluoromethyl 1H pyrrolo 2 3 b pyridine 3 carboxylic acid 5 fluoro 1H pyrazol 3 yl methanamine 6 aminoquinolin 2 1H one 1 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 chloro 5 nitro N phenylbenzamide 3 chloro 2 iodo 5 trifluoromethyl pyridine 2 bromo 4 fluoro 5 trifluoromethyl phenol 5 bromo 2 fluoropyridin 3 yl methanamine 3 fluorocyclobutan 1 ol 1 methyl 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 2 3 b pyridine 4 fluoro 1H pyrazolo 3 4 c pyridin 3 amine 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 2 fluoro 6 hydroxyphenylboronic acid 7 nitro 3 4 dihydronaphthalen 1 2H one 2 Bromo 6 fluorotoluene 2 3 dimethylbenzyl bromide