4 Fluoro 3 nitroacetophenone 2 Chloro 3 fluoropyridine 2 Bromo 3 fluorobenzoic acid 4 4 Hexafluoroisopropylidene diphthalic anhydride 1 3 5 Tris benzyloxy 1 3 5 triazinane 2 4 6 trione 2 Aminoacetophenone hydrochloride 2S 1 tert butoxy carbonyl 4 4 difluoro 2 methylpyrrolidine 2 carboxylic acid 3 methylidene 1 4 trifluoromethyl pyridin 2 yl cyclobutane 1 carbonitrile 5 fluoro 1H indole 7 carbonitrile 3 3 difluoro 2 oxoindoline 5 boronic acid pinacol ester 4 fluorobicyclo 2 2 1 heptane 1 carboxylic acid 2 2 difluoro 2H 1 3 benzodioxole 4 carbaldehyde 3 fluoro 1H pyrazole 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl naphthalen 2 amine 2 2 bromo 5 fluorophenyl propan 2 amine 4 methylpiperidin 4 ol 1 3 4 dichlorobenzyl indoline 2 3 dione 3 formylisonicotinonitrile 2 6 difluoro 4 methoxyphenol 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d thiazole 7 iodo 3 4 dihydronaphthalen 1 2H one 5 bromo 2 methylamino benzamide 2 Chloro 3 fluorophenyl isocyanate 6 fluoronaphthalen 2 ol 4 7 dichloro 1H indazole 4 bromo 1 methyl 1H indazole 2 3 difluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinonitrile 2 4 Dichloro 6 fluoro 3 nitrobenzoic acid 5 bromo 3 chloro 2 fluoronitrobenzene

3 Fluoro 4 morpholinylaniline 2 Chloro 6 fluorotoluene 7 Hydroxy 5 methyl 2 methylthio 1 2 4 triazolo 1 5 a pyrimidin 5 Fluoro 2 nitroanisole 2 Chloro 4 hydroxybenzaldehyde 2 4 Difluoroaniline 4 Bromo 2 chlorobenzyl bromide 2 3 Dichlorobenzyl alcohol 3 5 Difluoro 2 nitrobenzoic acid 2 5 DIFLUOROBENZOTRIFLUORIDE 5 Bromo 2 fluorophenylacetic acid 3 Bromo 4 methyl benzonitrile 3 Bromo 5 trifluoromethyl pyridin 2 ol 1 4 Cyclohexanedicarboxylic acid 3 4 5 Trimethoxybenzaldehyde 3 Trifluoromethyl phenylacetonitrile 3 Bromo 2 fluorobenzoic acid 4 4 HEXAFLUOROISOPROPYLIDENE DIPHTHALIC ACID 1 1 dithiodicarbonothioyl bis 1H Pyrazole 2 AMINO 5 BROMO 3 CHLOROPYRAZINE 2 trifluoromethoxy pyridin 4 amine 5 Bromo 1 methyl 3 trifluoromethyl 1H pyrazole 5 trifluoromethyl 1H indole 2 chloro N N diisobutylacetamide 3 amino 2 hydroxybenzenesulfonamide 4 4 nitro 1H pyrazol 1 yl piperidine 2 bromo 3 methoxyphenol 5 hydroxy 2 methylbenzonitrile 6 formylnicotinonitrile 2 4 morpholinomethyl phenyl acetic acid

6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d thiazole 2 6 dibromonicotinaldehyde 2 methoxy 5 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 3 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 fluoronaphthalen 2 amine 4 chloro 1H pyrazolo 3 4 b pyridine 7 bromo 1 methyl 1H indazole 2 Tert butyl phenyl isocyanate 2 Fluoro 4 methylsulfonyl aniline 3 Bromo 5 chloronitrobenzene 2 4 Dichloro 5 fluorobenzoyl chloride 3 bromo 5 chlorobenzamide 4 Methylaminopyridine 5 Hydroxy 3 4 dihydronaphthalen 1 2H one 2 Chloro 3 5 dibromo 6 fluorotoluene 3 Methyl 2 4 6 Tribromophenol 4 Fluoro 3 nitroanisole 5 Chloro 2 fluorobenzaldehyde 2 3 Difluoroaniline 3 5 Dibromobenzyl alcohol 1 3 Bis bromomethyl 5 methylbenzene 2 6 Difluoro 3 nitrobenzoic acid 4 Bromo 3 fluorophenylacetic acid 2 3 Difluorobenzotrifluoride 2 4 5 Trimethoxybenzaldehyde 2 Amino 4 nitrobenzoic acid 3 5 Dibromo 6 methylpyridin 2 amine 2 Hydroxy 1 8 naphthyridine 4 carboxylic acid 3 Fluoro 2 hydroxybenzaldehyde 2S 4 4 difluoropyrrolidine 2 carboxylic acid trifluoroacetic acid

3S 4S 1 tert butoxycarbonyl 3 fluoro piperidine 4 carboxylic acid 2 AMINO 5 TRIFLUOROMETHYL PYRAZINE 4 5 Difluoro 2 2 bis trifluoroMethyl 1 3 dioxole 5 Bromo 2 fluorobenzoic acid 2 2 difluoro 2 3 methyl 1H indazol 6 yl acetic acid 3 4 fluorophenyl azetidine hydrochloride 5 trifluoromethyl pyridine 3 carboxylic acid 7 fluoro 4 trifluoromethyl 1H indole 4 4 difluoropiperidin 3 ol hydrochloride 2 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 5 fluoro 3 4 dihydro 2H benzo b 1 4 oxazine 3 chloro 6 methoxypyridin 2 amine 6 bromo 2 iodoquinazoline 5 methylisoindoline 3 bromo 1 8 naphthyridine 3 chloro 4 methoxyphenol 4 bromo 2 3 dihydro 1H inden 1 one 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d thiazole 2 3 dichloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl picolinonitrile 6 bromo 1H pyrazolo 4 3 c pyridine 2 tert butoxycarbonylamino 3 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl propanoate 5 bromo 7 methyl 1H indazole 2 Chlorophenyl Isocyanate 2 Fluoro N methyl 5 nitroaniline 2 Bromo 4 chloro 1 iodobenzene 3 Trifluoromethyl benzamide 5 Methyl 2 tert butylphenol 2 Hydroxy 1 3 dihydro 2H isoindol 2 Methoxypyridine