2 4 6 Tribromopyrimidine 2 Morpholine 4 6 difluoropyrimidine 4 Bromo 2 fluoro 6 hydroxyacetophenone 4 Bromo 2 chloro 3 fluorophenol 4 Bromo propylbenzene 2 Fluoro 5 trifluoromethyl benzaldehyde 2 Chloro 4 methoxyacetophenone 2 Nitro 1 difluoromethoxy benzene 4 Chloro 3 fluorobenzyl chloride 4 Trifluoromethyl benzene 1 2 diamine 2 3 Trifluoromethyl phenyl ethanol 4 Nitro 2 trifluoromethyl benzoic acid 2 Nitro 4 trifluormethyl phenylacetic acid 2 fluoro 6 nitrotoluene 4 4 Diacetylbiphenyl 1 N boc pyrrolidin 2 ylboronic acid 4 Hydroxy 2 nitroanisole 4 Amino 2 6 dichlorophenol 3 Bromo 5 chloro 2 methoxypyridine 3 Fluoro 4 iodoaniline 2R 3S 2 2 4 difluorophenyl 3 5 fluoropyrimidin 4 yl 1 1H 1 2 4 triazol 1 yl butan 2 ol 4 N Boc AMinocyclohexanone 2 methyl 6 trifluoromethyl pyridine 3R 4R 4 fluoropyrrolidin 3 ol hydrochloride 2 fluoro 4 1H pyrazol 1 yl aniline 3 iodo 4 trifluoromethyl 1H pyrrolo 2 3 b pyridine 4 fluoro 1H indole 7 carbonitrile 1 azetidin 3 yl 3 fluoroazetidine oxalic acid 2 2 CARBOXYETHYL BENZOIC ACID 3 chloro 5 2 oxo 4 trifluoromethyl 1 2 dihydropyridin 3 yloxy benzonitrile

6 fluoroquinazolin 4 amine 3 chloro 4 dimethylcarbamoyl phenylboronic acid 3 4 dichloro N pentan 2 yl benzamide 5 bromo 2 ethylpyridine 1 2 bromo 6 methoxyphenyl ethanone 2 bromoquinolin 4 amine 4 nitrobenzene 1 3 diol 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 5 bromo 3 methyl 1H pyrazolo 4 3 b pyrazine 2 fluoro 5 hydroxyphenylboronic acid 3 Bromo 2 nitrotoluene 3 4 dihydro 2H benzo b 1 4 oxazin 8 ol 2 Amino 3 chlorobenzoic acid 3 5 Dibromo 2 methoxypyridine 4 4 Cyanophenyl phenol 5 Bromo 2 chloro 3 cyanopyridine 4 Butoxybiphenyl 2 6 Dibromopyridine 3 Nitrophenylacetic acid 3 Nitro 5 trifluoromethyl benzoic acid 2 Chloro 4 fluorobenzyl chloride 2 2 Trifluoromethyl phenyl ethanol 4 Methylbenzene 1 2 diamine 2 Fluoro 3 trifluoromethyl benzaldehyde 2 Chloro 6 hydroxyacetophenone 4 Nitro 1 2 chloroethoxy benzene 4 Bromo octylbenzene 2 Morpholine 4 6 dichloropyrimidine 4 Bromo 2 5 difluoroacetophenone 2 Bromo 4 chloro 6 fluorophenol

1 3 Diiodobenzene 2 Iodo 5 methoxybenzoic acid 3 Fluoro 5 iodobenzyl alcohol 3 Bromo 2 fluoropyridine 3 Fluoro 2 iodoaniline 4 4 Di tert butyl 2 2 bipyridine 4 5 dimethylquinolin 2 ol 3 bromo 4 trifluoromethyl 1H pyrrolo 2 3 b pyridine 3 trifluoromethyl 1H indol 6 amine hydrochloride 7 2 chloro 5 trifluoromethyl pyrimidin 4 yl amino 1 3 dihydro 2 1 benzoxaborol 1 ol 7 bromo 4 fluoro 1H indole 2 5 bromothiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 azetidin 3 yl 3 fluoroazetidine 2 4 fluorophenyl pyrrolidine 2 Methyloxazolo 4 5 b pyridine 5 amino 2 chloronicotinic acid 5 chlorothiazol 2 amine 4 fluoro 3 hydroxyphenylboronic acid 5 chloro 3 methyl 1H pyrazolo 4 3 b pyrazine 2 bromo 4 nitroquinoline 3 4 dimethoxy 2 nitrobenzaldehyde 2 bromo 6 hydroxybenzaldehyde 6 hydroxy 2H benzo b 1 4 oxazin 3 4H one 2 Fluoro 6 iodobenzyl alcohol 2 Bromo 6 nitrotoluene 2 4 Difluoro 1 3 5 trimethylbenzene 3 Bromo 4 chloroanisole 4 Methylphenyl diphenyl methanol 2’ 6’ Difluorophenacyl bromide 5 Nitrouracil

1 Methylthio 3 trifluoromethyl benzene 5 Bromo 2 iodo 1 3 diethylbenzene 4 Chloro 3 fluoroacetophenone 5 Fluoro 2 nitrobenzaldehyde 3 Methylbenzene 1 2 diamine 4 Chlorobenzyl chloride 2 4 Trifluoromethoxyl phenyl ethanol 2 Fluoro 4 iodoaniline 2 Bromo 5 trifluoromethyl pyridine 5 Amino 2 hydroxypyridine 4 Iodo 4 methylbiphenyl 1 Isopropenyl 4 methoxybenzene 1 3 Bis 2 4 6 trimethylphenyl 4 5 dihydroimidazol 2 ylidene 2 5 Dibromopyridine 4 Mercaptophenylacetic acid 3 Nitro 4 trifluoromethyl benzoic acid 4 4 Hydroxy 3 iodophenyl benzonitrile 4 2H benzo d 1 2 3 triazol 2 yl benzene 1 3 diol 5 fluoropyrazolo 1 5 a pyridine 1 cyclopropyl 6 7 difluoro 1 4 dihydro 4 oxo 1 8 naphthyridine 3 carboxylic acid 1h pyrrolo 3 2 b pyridine 5 carbonitrile 6 fluoro 3 trifluoromethyl 1H indol 6 amine 3 fluoro 4 morpholin 4 yl aniline 1 aminomethyl 4 4 difluorocyclohexan 1 ol 4 trifluoromethyl 1H pyrrolo 2 3 b pyridine 2 3 fluorophenyl pyrrolidine 5 chloro 6 iodoisoindolin 1 one 4 hydroxy N N 2 trimethyl 1 tosyl 1H benzo d imidazole 6 carboxamide 6 methoxy 5 trifluoromethyl pyridin 3 amine 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole