3 Tetrahydro 2H pyran 2 yloxy phenylboronic acid 2 Fluoro 5 isoproproxyphenylboronic acid 2 Ethoxy 5 methylphenylboronic acid 2 4 Dichloro 5 nitrophenylboronic acid 3 5 Dichloro 4 methoxyphenylboronic acid 2 Methoxycarbonylphenylboronic acid pinacol ester 3 Formylthiophene 2 boronic acid 4 Bromopyridine 3 boronic acid 3 Chloro 2 4 difluorophenylboronic acid 5 Chloro 2 4 difluorophenylboronic acid 4 N Butoxy 2 methylphenylboronic acid 3 Bromo 2 ethoxy 5 methylphenylboronic acid 4 Benzyloxy 3 5 dimethylphenylboronic acid 2 Benzyloxy 5 methylphenylboronic acid 3 Piperidine 1 carbonyl phenylboronic acid 4 Formyl 2 methylphenylboronic acid 3 Tetrahydro 2H pyran 2 yloxy phenylboronic acid pinacol ester 5 Formyl 2 ethoxyphenylboronic acid 3 Methylthiophenylboronic acid pinacol ester 4 Ethoxy 2 formylphenylboronic acid 2 4 Dimethoxyphenylboronic acid pinacol ester 2 3 Difluoro 4 n hexyloxy phenylboronic acid 2 Acetylaminophenylboronic acid pinacol ester 4 Aminocarbonyl phenylboronic acid pinacol ester 3 Benzyloxycarbonyl 5 nitrophenylboronic acid 2 Methoxy 4 methoxycarbonyl phenylboronic acid 2 Bromo 5 6 difluorophenylboronic acid 2 Bromo 3 ethoxy 6 fluorophenylboronic acid 2 Bromo 4 5 difluorophenylboronic acid 3 Bromo 2 fluorophenylboronic acid

4 Bromo 2 5 dimethoxyphenylboronic acid 1 Hexaneboronic acid cyclic iminodiethylene ester 2 Chloro 6 trifluoromethylbenzoic acid 3 Chloro 4 formylphenylboronic acid 3 Bromo 2 chloropyridine 4 boronic acid pinacol ester 4 Fluorophenylboronic acid pinacol ester 3 Cyano 4 5 5 Dimethyl 1 3 2 dioxaborinan 2 yl pyridine 2 Chloro 6 isopropylpyridine 3 boronic acid 4 Cyano 3 5 5 Dimethyl 1 3 2 dioxaborinan 2 yl pyridine 3 fluoro adamantane 1 methanol 5 6 chloropyridazin 3 yl methyl 2 2 fluorophenyl 5H imidazo 4 5 c pyridine 5 6 2 4 bis trifluoromethyl phenyl pyridazin 3 yl methyl 2 2 fluorophenyl 5H imidazo 4 5 c pyridine 3 difluoromethylpiperidine hydrochloride 4 Hydroxydibenzothiophene 1 4 2 4 difluorobenzoyl piperidin 1 yl 2 2 2 trifluoroethanone 1 1 benzylpiperidin 4 yl 2 2 2 trifluoroethanone oxalate 4 4 difluoropiperidin 3 ol hydrochloride 2 2 2 trifluoro 1 4 4 fluorobenzoyl piperidin 1 yl ethanone 1 1 piperidine 1 4 diyl bis 2 2 2 trifluoroethanone 3 FLUOROPIPERIDINE HYDROCHLORIDE 1 tert butoxycarbonyl 5 5 difluoropiperidine 2 carboxylic acid 2 3 difluoro 4 nitrophenol 3 amino 2 2 difluoropropanoic acid hydrochloride 3 3 difluoro 5 hydroxypiperidin 2 one 1 tert butoxycarbonyl 5 5 difluoropiperidine 3 carboxylic acid 1 2 2 2 TRIFLUOROACETYL 4 PIPERIDINECARBOXYLIC ACID 4 fluoro 2 methylamino benzoic acid 1 tert butoxycarbonyl 3 3 difluoropiperidine 4 carboxylic acid 1 tert butyl 3 methyl 4 4 difluoropiperidine 1 3 dicarboxylate 3 4 cis 1 benzyloxycarbonyl 3 fluoropiperidine 4 carboxylic acid

1 tert butoxycarbonyl 4 4 difluoropiperidine 3 carboxylic acid 4 4 DIFLUOROADAMANTANE 1 CARBOXYLIC ACID METHYL ESTER 1 benzyl 3 difluoromethylene piperidine 1 benzyl 4 fluoropiperidin 3 yl methyl acetate 1 tert butyl 3 ethyl 5 5 difluoro 4 oxopiperidine 1 3 dicarboxylate 2 1 tert butoxycarbonyl 3 fluoropiperidin 4 yl acetic acid 4 Trifluoroacetyl piperidine hydrochloride 1 tert butyl 4 ethyl 5 fluoro 4 methyl 3 4 dihydropyridine 1 4 2H dicarboxylate 3 acetamido 6 acetyl 2 nitrophenyl 4 dimethylamino 3 5 difluorobenzoate 1 tert butyl 3 ethyl 5 fluoropiperidine 1 3 dicarboxylate 4 trifluoromethyl 1 4 5 6 tetrahydropyridine 3 carbonitrile 2 2 2 trifluoro 1 4 4 bromobenzoyl piperidin 1 yl ethanone 2 2 2 trifluoro 1 4 benzoylpiperidin 1 yl ethanone 2 2 trifluoromethoxy ethyl isoindoline 1 3 dione 4 fluoromethylpiperidine hydrochloride 4 4 4 trifluoro 1 3 methoxyphenyl butane 1 3 dione 4 4 DIFLUOROADAMANTANE 1 CARBOXYLIC ACID 1 tert butoxycarbonyl 4 fluoropiperidine 4 carboxylic acid 1 tert butyl 4 ethyl 4 4 fluorobenzyl piperidine 1 4 dicarboxylate with Methy ester analog 1 Trifluoromethyl 1 2 benziodoxol 3 1H one 4 difluoromethyl piperidine hydrochloride 4 tert butoxycarbonylamino 3 3 difluorobutanoic acid 4 1 Hydroxy 2 2 2 trifluoroethyl piperidine oxalate 2S 4S 1 tert butyl 2 methyl 4 fluoropyrrolidine 1 2 dicarboxylate 2 2 fluorophenyl 3H imidazo 4 5 c pyridine methanesulfonate 3 2 2 4 dimethylphenyl 2 2 2 2 trifluoroacetyl hydrazono methyl benzoic acid 3R 4S tert butyl 3 fluoro 4 R 1 4 methoxyphenyl ethylcarbamoyl piperidine 1 carboxylate enantiomer a e e 95 4 benzyl 3 3 difluoropiperidine hydrochloride 2 1 tert butoxycarbonyl 4 4 difluoropiperidin 3 yl acetic acid 1 tert butoxycarbonyl 4 4 fluorobenzyl piperidine 4 carboxylic acid

1 benzyl 3 3 difluoro 4 phenylpiperidin 4 ol 3 3 difluoro 4 phenylpiperidine hydrochloride 5 azidomethyl 3 3 difluoro dihydrofuran 2 3H one 4 4 difluoropiperidin 3 yl methanol hydrochloride 3 4 cis tert butyl 4 azido 3 fluoropiperidine 1 carboxylate 3 4 trans tert butyl 4 azido 3 fluoropiperidine 1 carboxylate 3 4 trans 1 benzyloxycarbonyl 3 fluoropiperidine 4 carboxylic acid 2 1 tert butoxycarbonyl 3 3 difluoro 1 2 3 6 tetrahydropyridin 4 yl acetic acid 5 Methoxy 2 phenylbenzonitrile 5 benzyl 7 7 difluoro 4 5 6 7 tetrahydroisoxazolo 4 5 c pyridin 3 ol 6 Bromo 2 fluoro 3 iodobenzaldehyde 3 4 Trans 1 tert butoxycarbonyl 3 fluoropiperidine 4 carboxylic acid racemate 6 Bromo 2 chloro 3 methylbenzoic acid 3R 4S 1 tert butoxycarbonyl 3 fluoropiperidine 4 carboxylic acid enantiomer a 95 e e 4 Bromo 3 chlorobenzyl alcohol 3 4 Cis tert butyl 3 fluoro 4 hydroxymethyl piperidine 1 carboxylate 2 Bromo 5 methylphenyl methanol 1 tert butyl 3 ethyl 5 5 difluoro 5 6 dihydropyridine 1 3 2H dicarboxylate 2 6 Difluoro 3 methylthio benzyl alcohol 3 Bromo 2 fluoro 5 trifluoromethyl benzaldehyde 3 Bromo 4 methylbenzyl alcohol 3 5 Dibromo 4 methoxyphenyl methanol 3 4 Tras tert butyl 3 fluoro 4 hydroxymethyl piperidine 1 carboxylate 2 Bromo 6 fluoro 3 trifluoromethyl benzaldehyde 4 Bromo 2 methoxybiphenyl 3 Chloro biphenyl 4 ylamine 3 Methylthio 5 trifluoromethyl benzoic acid 2 Bromo 5 iodobenzyl alcohol 2 Amino 5 trifluoromethoxy biphenyl 2 Chloro 4 isopropoxybenzaldehyde