4 Ethynylquinoline 2 6 Bromopyridin 3 yl pyrimidine 1 3 Fluorobenzyl 5 oxo pyrrolidine 3 carboxylic acid 7 Bromo 1 2 4 triazolo 1 5 a pyridine 3 Methylazetidine hydrochloride 1 Methyl 1H indazol 5 ol 4 Bromo 6 methylpyrimidine 4 Methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 2 4 Fluorophenyl 2 3 dihydro 4 1H quinolinone 2 Thiazole acetic acid 3 4 Fluorophenyl phenethyl alcohol 1 Methyl 2 methylthio 4 5 dihydro 1H imidazole hydroiodide 6 Bromo N N dimethyl 2 quinazolinamine 1 Methyl 4 nitroimidazole 6 Chloro 4 pyridazinamine 1 Methyl 1H pyrazole 4 sulfonyl chloride 6 Bromo 8 methoxyimidazo 1 2 a pyrazine 2 Methoxy 4 4 methylpiperazin 1 yl aniline 4 Bromobenzo d isoxazole 2 3 Chloro 5 trifluoromethyl phenyl acetonitrile 2 4 Dihydroxypteridine 7 Bromo 1 2 4 triazolo 1 5 a pyridin 2 amine 6 Bromo 3 iodoimidazo 1 2 a pyrazine 5 Ethynyl 3 methyl 1H indazole 4 Hydroxypyrimidine 5 carboxylic acid 4 Pyridin 3 yloxy benzoic acid 2 4 Dichloro 5 7 dihydrofuro 3 4 d pyrimidine 2 5 6 Trichloro 4 methyl 3 pyridinecarbonitrile 1R 4S 7 Boc 2 oxo 7 azabicyclo 2 2 1 heptane 3 Fluoropyrrolidine hydrochloride

2 Bromobenzo d thiazole 6 carbonitrile 3 Amino 6 chloro 2 pyrazinecarbonitrile 1 Aminomethyl cyclobutanol 4 Chloro 3 methyl 1H pyrrolo 2 3 b pyridine 1 2 4 Triazolo 4 3 a pyrazine 3 carboxylic acid 1 4 Bromophenyl cyclobutanamine hydrochloride 6 Bromoquinoline 4 carboxylic acid 6 Benzyloxy pyridine 2 carboxylic acid 6 Chloro 2 methyl 1H indole 3 Amino 1H pyrazol 5 ol 4 Benzyloxy 2 6 difluorophenylboronic acid 5 chloro 4 fluoro 2 nitrophenol 1H pyrazolo 4 3 c pyridine 3 carboxylic acid 6 Bromo 3 hydroxypicolinic acid 4 Chloro 6 isopropoxypyrimidine 1 Boc 3 iodo 1H indazole 7 Bromo 1 2 dihydroisoquinolin 3 4H one 5 Iodo 4 methylpyrimidine 6 Bromo 1 2 4 triazolo 1 5 a pyrazine 2 Chloro 6 nitroquinoxaline 2 Amino 4 morpholin 4 yl pyrimidine 6 Chloro N methyl 5 nitro 4 pyrimidinamine 1 Boc 5 6 Dichloro 1H indole 3 Bromoimidazo 1 2 b pyridazin 6 ylamine 1 Boc 4 Cbz aminoazepane 8 Chloro 2 methylimidazo 1 2 a pyrazine 6 8 Dibromo 1 2 4 triazolo 1 5 a pyrazine 2 Methylsulfonyl pyrimidine 4 carboxylic acid 2 4 Methylpiperazin 1 yl pyrimidin 5 amine 5 Bromo 2 cyanobenzeneacetonitrile

5 Bromo 4 chloropyrimidin 2 amine 7 Bromoisoquinolin 3 amine 3 3 Fluorophenoxy methyl piperidin 3 ol 7 Fluoroquinoline 6 carbaldehyde 3 tert butyl 1H pyrazol 4 carbaldehyde 6 Bromo 1H indazole 4 carboxylic acid 5 Amino 2 fluoro 4 nitrobenzotrifluoride 4 Bromo 2 chloro 3 fluorophenol 2 6 Dichloro 3 nitrobenzoic acid 3 Fluoro 4 methyl 5 hydroxybenzoic acid 4 3 Bromoimidazo 1 2 b pyridazin 6 yl morpholine 7 Bromothieno 2 3 b pyrazine 8 Bromoisoquinolin 1 2H one 4 Methyltetrahydro 2H pyran 4 ol 4 Bromo 2 cyanobenzeneacetonitrile 5 Ethynylpyrimidine 1 Pyridazin 4 yl ethanone 5 Bromo 3 fluoropyridin 2 amine 2 Amino 5 bromo 3 chloropyrazine 4 1 Piperazinyl 6 trifluoromethyl pyrimidine 7 Nitro 2 1H quinoxalinone 2 Chlorothiazol 5 yl methylamine hydrochloride 5 Bromo 2 chlorobenzyl amine 2 hydroxy 4 methylthiazole 5 carboxylicacid 7 Fluoro 1H indole 2 carboxylic acid 3 5 Dimethylpyrazin 2 ol 5 Bromo N methylpyrimidin 4 amine 4 5 Dichloropyrimidin 2 amine 5 Methyl 3 nitro 1H pyrazole 4 Flurophenyl acetic acid ethyl ester

5 Chloro 1 3 4 thiadiazol 2 amine 2 3 Dibromopyrazine 2 3 4 5 Tetrahydro 1H benzo c azepine hydrochloride 1R 2S 2 Aminocyclohexanol hydrochloride 4 2 Bromoethyl benzonitrile 4 1 Pyrrolidinyl 3 trifluoromethyl bezenamine dihydrochloride 2 2 4 Dichlorophenyl thiazole 4 carboxylic acid 2 Chloro 4 morpholinothieno 3 2 d pyrimidine 6 carbaldehyde 6 Bromochromen 2 one 2 4 Dichloro 5 6 7 8 tetrahydropyrido 4 3 d pyrimidine hydrochloride 3 Phenyl 3 pentylamine hydrochloride 3 Amino 2 fluorophenyl methanol 4 Amino N methylbenzeneethanesulfonamide 1 Piperidin 4 yl pyrrolidin 2 one 4 Amino 6 iodopyrimidine 2 Chloro 5 isopropylpyrimidine 4 Chloro 7 trifluoromethyl quinazoline 4 Methylamino 3 nitropyridine 6 Hydroxyimidazo 1 2 b pyridazine 1 Boc 3 Cyano 4 hydroxypyrrolidine 4 Chloro 6 trifluoromethyl 1H pyrazolo 3 4 d pyrimidine 2 4 Methyl 1 piperazinyl 4 pyrimidinamine 1 2 3 4 Tetrahydropyrido 2 3 b pyrazine 2 Amino 3 methoxybenzaldehyde 1 Boc 3 Iodo 7 azaindole 2 4 Bromo 1H pyrazol 1 yl pyrimidine 2 Amino 6 bromopyrido 2 3 d pyrimidin 4 3H one 3 4 Bromopyrazol 1 ylmethyl pyridine 6 Hydroxy 1 2 benzisoxazole 1 Boc 5 Bromo 1 2 dihydro 2 oxo spiro 3H indole 3 4 piperidine