2 3 Dimethyl 4 methoxyphenylboronic acid 2 Chloro 5 formylphenylboronic acid pinacol ester 5 chloro 2 fluoro 3 4 4 5 5 tetramethyl 1 3 dioxolan 2 yl pyridine 4 Biphenyl 4 yl piperidine 4 Bromo 2 5 bifluorophenylboronic acid pinacol ester 2 Chloro 6 hydroxyphenylboronic acid pinacol ester 2 6 Difluoro 3 methylthio phenylboronic acid 1 tert butyl 4 ethyl 3 hydroxy 4 methylpiperidine 1 4 dicarboxylate 4 Ethoxy 2 3 dimethylphenylboronic acid 1 tert butoxycarbonyl 1 2 3 6 tetrahydropyridine 4 carboxylic acid 2 8 tert butoxycarbonyl 8 aza bicyclo 3 2 1 octan 3 yl acetic acid 2 Fluoro 4 methoxycarbonyl phenylboronic acid pinacol ester 2 6 Dimethyl 4 fluorophenylboronic acid 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 6 tetrahydropyridine 1 benzyl 3 methyl 5 tert butoxycarbonylamino piperidine 1 3 dicarboxylate 4 Cyano 3 methylphenylboronic acid pinacol ester 4 Bromo 2 methylphenyboronic acid 4 Fluoro 1H indazol 6 yl boronic acid 3 bromo 1 propyl 1 2 5 6 tetrahydropyridine 3 Bromophenylboronic acid N butyldiethanolamine ester 2 Trifluoromethylpyridine 5 boronic acid pinacol ester 4 Bromo 2 isopropylphenylboronic acid 3 Bromo 5 formylphenylboronic acid 2 8 DIAZASPIRO 5 5 UNDECAN 1 ONE HYDROCHLORIDE 4 5 Amino 1H pyrazol 3 yl piperidine 1 carboxylic acid tert butyl ester 3 Bromo 4 chlorophenylboronic acid 3 hydroxy 4 5 6 7 tetrahydro 2H pyrazolo 3 4 c pyridine 5 carboxylic acid hydrochloride 4 4 bromophenyl piperidine 4 carbonitrile 4 Methoxy 2 trifluoromethoxy phenylboronic acid 2 Fluoro 4 formyl 6 methoxyphenylboronic acid

2 4 Difluoro 3 iodophenylboronic acid 6 Isobutoxy 2 methylpyridine 3 boronic acid 7 Chloro 1H indazole 4 boronic acid 2 Bromo 4 methylphenylboronic acid 1 benzyl 4 3 phenylpropyl 1 2 3 6 tetrahydropyridine 3 5 Dichloro 2 6 difluorophenylboronic acid 1 benzyl 3 1 benzyl 2 oxo piperidin 4 ylidene piperidine 2 4 dione 6 Isopropoxynaphthalene 2 boronic acid 1 tert butyl 2 ethyl 3 oxopiperidine 1 2 dicarboxylate 3 3 difluoropiperidin 4 ol 6 Isopropoxy 2 methylpyridine 3 boronic acid 2 3 Dimethoxypyridine 5 boronic acid 2 Fluoro 3 isopropoxypyridine 5 boronic acid 5 Fluoro 2 morpholin 4 ylmethyl phenyl boronic acid 5 Chloro 2 methylsulfanyl pyridine 3 boronic acid 1 tert butyl 3 methyl 5 oxopiperidine 1 3 dicarboxylate 4 Bromo 2 Chloro 5 trifluoromethyl phenylboronic acid 3 Bromo 5 methylsulfanyl phenylboronic acid 4 Bromo 2 fluoro 5 trifluoromethyl phenylboronic acid 2 Ethoxy 4 methylphenylboronic acid 4 Bromo 5 chloro 2 methylphenylboronic acid 1 HYDROXYMETHYL 3 OXO 2 AZABICYCLO 2 2 2 OCTANE 2 Chloro 3 5 dimethylphenylboronic acid 2 6 Dimethoxybiphenyl 2 ylboronic acid 1 benzyl 3 hydroxymethyl piperidin 4 ol 4 Amino 3 5 dimethylphenylboronic acid pinacol ester 4 Chloro 3 isopropoxyphenylboronic acid 2 Fluoro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid methyl ester 8 benzyl 3 hydroxyimino 8 AZA BICYCLO 3 2 1 OCTANE 2 Amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile

2 Tert butylcarbonylamino phenylboronic acid pinacol ester 8 benzyl 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octane 2 Phenoxypyridine 5 boronic acid 6 Fluoro 2 methylsulfanyl phenylboronic acid 2 Bromo 4 chlorophenylboronic acid 4 4 bromophenyl piperidine 4 carbonitrile hydrochloride 5 tert butyl 3a ethyl hexahydro 1H pyrrolo 3 2 c pyridine 3a 5 6H dicarboxylate 5 Fluoro 2 morpholinomethyl phenylboronic acid hydrochloride 1 methyl 4 phenylpiperidine 2 Methoxy 4 methylthio pyridine 5 boronic acid 2 Methoxy 4 methylthio pyridine 5 boronic acid pinacol ester 4 Isopropoxy 3 trifluoromethyl phenylboronic acid 4 Fluoro 3 methanesulfonyl phenylboronic acid 2 Methylthio thiophene 3 boronic acid 2 Methylthio thiophene 4 boronic acid 3 Methoxy 2 methylphenylboronic acid 2 CHLORO 3 METHYL 5 PHENYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 3 Bromo 5 carboxythiophene 2 boronic acid 2 CHLORO 3 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 4 N Boc piperazino pyridine 5 boronic acid 2 Benzyloxy 4 methylpyridine 5 boronic acid 2 TRIFLUOROMETHYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 3 Bromo 2 formylthiophene 5 boronic acid 3 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 3 PYRIDINAMINE 2 Phenoxypyridine 4 boronic acid 2 CHLORO 5 METHOXYPYRIDINE 4 BORONIC ACID 2 Isopropoxy 4 methylpyridine 5 boronic acid pinacol ester 2 CARBOXYPYRIDINE 4 BORONIC ACID 2 Isopropoxy 4 methylpyridine 5 boronic acid

5 BROMO 2 TRIFLUOROMETHYL PYRIDIN 4 YLBORONIC ACID 4 Benzyloxy 2 chlorophenylboronic acid 6 Ethoxy 2 fluoro 3 methylphenylboronic acid 2 CHLORO 3 FLUORO 5 PICOLINE 4 BORONIC ACID 5 Methyl 1H indazole 4 boronic acid 2 TRIFLUOROMETHYL PYRIDINE 4 BORONIC ACID 2 4 Difluoro 3 hydroxymethyl phenylboronic acid 4 Piperazin 1 ylmethyl phenylboronic acid 2 CHLORO 3 FLUOROPYRIDINE 4 BORONIC ACID 4 BORONO 2 6 PYRIDINEDICARBOXYLIC ACID 2 6 DIETHYL ESTE 4 2 methylpropyl amino methyl phenylboronic acid 6 Fluoro 2 hydroxy 3 methylphenylboronic acid pinacol ester 2 N BOC AMINO 6 ETHOXYCARBONYL 4 PYRIDINE BORONIC ACID PINACOL ESTER 3 4 Dichloropyridine 5 boronic acid pinacol ester 4 Bromo 3 fluorophenylboronic acid pinacol ester 1 3 DIHYDRO 1 HYDROXY 1 2 OXABOROLO 4 3 C PYRIDINE 2 Fluoro 4 morpholinomethyl phenylboronic acid 2 CYANOPYRIDIN 4 YL BORONIC ACID 5 Hydroxymethylthiophene 2 boronic acid pinacol ester 2 HYDROXY PYRIDINE 4 BORONIC ACID 2 Fluoro 4 morpholinomethyl phenylboronic acid pinacol ester 2 TERT BUTYLDIMETHYLSILYLOXY METHYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 3 N N Dimethylaminomethyl phenylboronic acid pinacol ester 2 CHLORO 3 CYANOPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 Fluoro 4 5 dimethoxyphenylboronic acid 5 BROMO 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 2 PYRIDINECARBONITRILE 5 Diethylamino methyl 2 fluorophenylboronic acid 2 6 DIMETHYL PYRIDINE 4 BORONIC ACID 2 4 Difluoro 3 isopropoxyphenylboronic acid 4 Isobutoxyphenylboronic acid