1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl morpholine 1 methyl 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 2 chloro 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 propoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 fluoro 1H indazole 6 carboxylic acid 3 methyl 1H indazol 7 amine 5 chloro 3 trifluoromethyl 1H indazole 3 bromo 6 trifluoromethyl 1H indazole 3 iodo 6 trifluoromethyl 1H indazole 6 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 2 amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinic acid 2 3 dimethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrido 2 3 b pyrazine 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 3 2 b pyridine 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinonitrile 2 methoxy 5 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 chloro 2 isopropoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 ethoxy 6 methylpyridin 3 yl boronic acid 2 piperidin 1 yl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 chloro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 4 fluoro 3 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 4 dimethylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 methoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 2 fluoro 5 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 chloro 6 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 fluoro 3 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 5 chloro 2 methoxymethoxy phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 fluoro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl ethanol

2 3 chloro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 fluoro 3 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl ethanol 4 4 5 5 tetramethyl 2 perfluorophenyl 1 3 2 dioxaborolane 4 4 5 5 tetramethyl 2 2 3 4 trifluorophenyl 1 3 2 dioxaborolane 2 fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 2 fluoro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 4 chloro 2 6 difluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 4 chloromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 chloro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 hydroxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 trifluoromethyl phenol 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl phenol 5 fluoro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 3 difluoro 4 methylphenyl boronic acid 3 4 bis methoxycarbonyl phenyl boronic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d 1 2 3 triazole 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d 1 2 3 triazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl indoline 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indole 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 ol 2 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 2 5 methoxynaphthalen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoindolin 1 one 2 hydroxy 5 trifluoromethyl phenyl boronic acid 2 hydroxy 4 trifluoromethyl phenyl boronic acid 4 fluoro 2 hydroxyphenyl boronic acid

5 borono 2 hydroxybenzoic acid 4 hydroxy 2 methylphenyl boronic acid 3 chloro 5 fluoro 4 methoxyphenyl boronic acid 2 chloro 5 fluorophenyl boronic acid 3 chloro 4 cyanophenyl boronic acid 4 5 difluoro 2 hydroxyphenyl boronic acid 3 5 difluoro 2 hydroxyphenyl boronic acid 3 fluoro 4 hydroxyphenyl boronic acid 2 hydroxy 5 methoxyphenyl boronic acid 3 chloro 4 hydroxyphenyl boronic acid 2 chloro 5 methoxyphenyl boronic acid 4 cyano 3 5 difluorophenyl boronic acid 4 fluoro 2 methoxyphenyl boronic acid 2 4 dichloro 6 fluorophenyl boronic acid 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 3H one 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 3H one 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 2 3 dimethyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyrimidine 7 methylimidazo 1 2 a pyridin 6 yl boronic acid 7 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 1 methyl 1H indazol 7 yl boronic acid 1H indazol 7 yl boronic acid 1H indazol 4 yl boronic acid 1H indazol 5 yl boronic acid 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 3 amine 3 methylsulfonyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinaldehyde

5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl methanol 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl ethanone 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methanol 3 butoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 ethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 4 5 5 tetramethyl 2 3 methylbenzofuran 6 yl 1 3 2 dioxaborolane 7 methylbenzofuran 5 yl boronic acid 2 7 chlorobenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 benzo b thiophen 3 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 hydroxymethyl thiophen 2 yl boronic acid 3 bromothiophen 2 yl boronic acid 3 methylthiophen 2 yl boronic acid 4 bromo 5 methylthiophen 2 yl boronic acid 2 5 chlorothiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 4 chlorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 4 fluorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 3 chlorophenyl 1H pyrazol 4 yl boronic acid 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 4 fluorophenyl 1H pyrazol 4 yl boronic acid 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl morpholine 2 piperidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl propan 2 ol 2 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 carbonitrile 4 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 ethoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 isopropoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine