3 borono 5 methoxybenzoic acid 4 methoxy 2 trifluoromethyl phenyl boronic acid 2 chloro 4 cyanophenyl boronic acid 2 chloro 4 methoxyphenyl boronic acid 2 6 dimethoxyphenyl boronic acid 2 cyano 5 methoxyphenyl boronic acid 2 chloro 4 fluorophenyl boronic acid 3 methoxy 5 trifluoromethyl phenyl boronic acid 5 ethyl 2 hydroxyphenyl boronic acid 4 5 difluoro 2 methoxyphenyl boronic acid 3 ethylbenzene 1 2 diol 3 chloro 5 fluorophenol 4 chloro 2 hydroxyphenyl boronic acid 2 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 4 tetrahydroisoquinoline 2 chloro 4 methoxyphenol 2 fluoro 5 methylphenol 4 methoxy 3 methylphenol 4 tert butyl 2 hydroxyphenyl boronic acid 1 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 3 4 dihydroisoquinolin 2 1H yl ethanone 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoxalin 2 ol 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 8 trifluoromethyl quinoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d thiazole 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H imidazo 4 5 b pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 2 3 b pyridin 2 3H one 4 4 5 5 tetramethyl 2 7 trifluoromethyl benzo b thiophen 2 yl 1 3 2 dioxaborolane 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 1 yl ethanone 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyrimidine 8 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 trityl 1H pyrazolo 3 4 b pyridine 2 5 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane

2 7 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 4 5 5 tetramethyl 2 5 methylbenzo b thiophen 2 yl 1 3 2 dioxaborolane 4 4 5 5 tetramethyl 2 3 methylbenzo b thiophen 5 yl 1 3 2 dioxaborolane 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazol 2 yl morpholine 2 cyclohexyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 2 isopropyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 trityl 1H pyrazole 1 4 methoxybenzyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 3 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl pyridine 1 methyl 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl piperidine 2 methyl 1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl propan 2 ol 1 2 methoxyethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 isopentyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 4 diethoxypyrimidin 5 yl boronic acid 1 cyclopropyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 tert butyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 6 dimethoxypyrimidin 5 yl boronic acid 2 1H imidazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl piperidin 4 one 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl piperidin 4 ol 3 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 piperazin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 3 propoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 isopropoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 4 methoxyaniline 2 butoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methylsulfonyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methanamine 2 propoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine

1 isopentyl 1H pyrazol 4 yl boronic acid 1 ethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 trityl 1H pyrazol 4 yl boronic acid 1 methyl 1H pyrazol 4 yl boronic acid 1 isobutyl 1H pyrazol 4 yl boronic acid 1 benzyl 1H pyrazol 4 yl boronic acid 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 2 isopropoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl pyridin 2 amine 2 4 methyl 1H pyrazol 1 yl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 1 1 diethoxyethyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methylthio 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 benzyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 1H one 1 3 dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 1H one 6 methyl 1H pyrazolo 3 4 b pyridine 3 bromo 6 chloro 1H pyrazolo 3 4 b pyridine 6 chloro 3 trifluoromethyl 1H pyrazolo 3 4 b pyridine 3 chloro 1H indazol 5 amine 3 bromo 6 nitro 1H indazole 5 bromo 3 chloro 1H indazole 4 bromo 3 iodo 1H indazole 4 bromo 3 chloro 1H indazole 4 chloro 3 iodo 1H indazole 3 bromo 5 chloro 1H indazole 5 chloro 3 iodo 1H indazole 7 chloro 3 iodo 1H indazole 3 bromo 7 fluoro 1H indazole 3 bromo 4 fluoro 1H indazole 6 bromo 3 iodo 1H indazole 5 chlorothieno 2 3 b pyridine

7 chlorothieno 2 3 c pyridine 5 chlorothieno 2 3 c pyridine 4 chloro 3 methylbenzo b thiophene 5 chloro 3 methylbenzo b thiophene 3 methoxy 2 nitroaniline 6 chloro 3 methylbenzo b thiophene 5 bromo 1H pyrazolo 4 3 b pyrazin 3 amine 5 iodo 1H pyrazolo 4 3 b pyrazin 3 amine 5 bromo 1H pyrazolo 4 3 b pyrazine 5 bromo 3 methyl 1H pyrazolo 4 3 b pyrazine 5 chloro 1H pyrazolo 4 3 b pyrazine 5 chloro 3 methyl 1H pyrazolo 4 3 b pyrazine 3 bromo 1H pyrazolo 4 3 b pyrazine 4 bromo 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 5 chloro 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 4 chloro 1H pyrazolo 3 4 c pyridin 3 amine 4 fluoro 1H pyrazolo 3 4 c pyridin 3 amine 7 chloro 5 trifluoromethyl 1H pyrazolo 3 4 c pyridine 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 6 bromo 1H pyrazolo 4 3 b pyridin 3 amine 6 bromo 1H pyrazolo 4 3 b pyridine 7 chloro 1H pyrazolo 4 3 b pyridine 5 bromo 1H pyrazolo 4 3 b pyridin 3 amine 4 bromo 1H pyrazolo 4 3 c pyridin 3 amine 6 methyl 1H pyrazolo 3 4 b pyridin 3 amine 2 6 dimethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 butoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinaldehyde 2 fluoro 4 iodo 6 methoxypyridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 6 trifluoromethyl pyridine