5 chloro 1H pyrazolo 4 3 b pyrazine 5 chloro 3 methyl 1H pyrazolo 4 3 b pyrazine 5 bromo 3 methyl 1H pyrazolo 4 3 b pyrazine 3 bromo 1H pyrazolo 4 3 b pyrazine 4 fluoro 1H pyrazolo 3 4 c pyridin 3 amine 4 bromo 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 4 chloro 1H pyrazolo 3 4 c pyridin 3 amine 7 chloro 5 trifluoromethyl 1H pyrazolo 3 4 c pyridine 5 chloro 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 2 6 dimethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 methyl 1H pyrazolo 3 4 b pyridin 3 amine 4 bromo 1H pyrazolo 4 3 c pyridin 3 amine 5 bromo 1H pyrazolo 4 3 b pyridin 3 amine 6 bromo 1H pyrazolo 4 3 b pyridin 3 amine 6 bromo 1H pyrazolo 4 3 b pyridine 7 chloro 1H pyrazolo 4 3 b pyridine 2 fluoro 4 iodo 6 methoxypyridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 6 trifluoromethyl pyridine 2 pyrrolidin 1 yl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinaldehyde 2 butoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 isobutoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 6 diethoxypyridin 3 yl boronic acid 3 1H imidazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 methyl N 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl benzenesulfonamide 3 fluoro N methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinonitrile 2 chloro 5 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl picolinonitrile

2 fluoro 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 ol 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 5 naphthyridine 3 bromo 7 trifluoromethyl 1H indazole 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 2 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 2 2 methoxy 5 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 methoxy 3 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 chloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 1 3 dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 4 1H 3H dione 3 trifluoromethyl 1H indazol 6 ol 3 methyl 4 nitro 1H indazole 3 methyl 5 nitro 1H indazole 4 4 5 5 tetramethyl 2 2 methyl 5 trifluoromethyl phenyl 1 3 2 dioxaborolane 2 2 6 difluoro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 2 4 dichloro 6 fluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 dichloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 2 5 chloro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 difluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 2 chloro 5 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 chloro 5 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 2 chloro 3 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 chloro 6 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 3 5 difluoro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 fluoro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 fluoro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile

4 4 5 5 tetramethyl 2 2 4 6 trichlorophenyl 1 3 2 dioxaborolane 2 2 chloro 5 fluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 4 tert butyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 chloro 5 fluoro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 chloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 fluoro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 3 5 difluoro 4 methoxycarbonyl phenyl boronic acid 2 tert butyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 3 cyano 2 4 difluorophenyl boronic acid 3 4 dimethylphenyl boronic acid 1 4 boronophenyl cyclopropanecarboxylic acid 4 1 methoxycarbonyl cyclopropyl phenyl boronic acid 4 hydroxy 2 trifluoromethyl phenyl boronic acid 2 6 difluoro 4 methoxyphenyl boronic acid 4 fluoro 3 methoxyphenyl boronic acid 2 methoxy 3 trifluoromethyl phenyl boronic acid 4 chloro 2 3 difluorophenyl boronic acid 2 fluoro 5 methylphenyl boronic acid 5 chloro 2 methoxyphenyl boronic acid 2 chloro 3 methoxyphenyl boronic acid 5 chloro 2 methoxymethoxy phenyl boronic acid 2 fluoro 4 methoxyphenyl boronic acid 3 chloro 5 fluoro 4 hydroxyphenyl boronic acid 3 chloro 5 fluorophenyl boronic acid 2 chloro 5 hydroxyphenyl boronic acid 2 fluoro 4 hydroxyphenyl boronic acid 2 hydroxy 4 methylphenyl boronic acid 2 hydroxy 5 methylphenyl boronic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzofuran 3 2H one

6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinolin 4 ol 1 chloro 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoquinoline 2 3 dihydrobenzofuran 4 yl boronic acid 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 amine 8 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazol 2 amine 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 amine 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 amine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 3 amine 1H indazol 6 yl boronic acid 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 7 trifluoromethyl 1H indazole 3 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 3 methyl 1H indazol 5 yl boronic acid 3 methyl 1H indazol 6 yl boronic acid 6 fluoro 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 1 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 1 methyl 1H indazol 4 yl boronic acid 3 methylthio 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 methoxymethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinamide 4 4 5 5 tetramethyl 2 3 methylbenzofuran 5 yl 1 3 2 dioxaborolane 2 6 chlorobenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 7 chlorobenzofuran 6 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 6 fluorobenzo b thiophen 7 yl boronic acid 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiophen 2 yl ethanone 4 methoxypicolinaldehyde