3 methylsulfonyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 methyl 1H indazol 7 yl boronic acid 1H indazol 7 yl boronic acid 1H indazol 4 yl boronic acid 1H indazol 5 yl boronic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinaldehyde 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl methanol 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl ethanone 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methanol 3 butoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 ethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 4 5 5 tetramethyl 2 3 methylbenzofuran 6 yl 1 3 2 dioxaborolane 3 methylthiophen 2 yl boronic acid 4 bromo 5 methylthiophen 2 yl boronic acid 3 bromothiophen 2 yl boronic acid 3 hydroxymethyl thiophen 2 yl boronic acid 2 benzo b thiophen 3 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 7 chlorobenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 7 methylbenzofuran 5 yl boronic acid 2 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 2 5 chlorothiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 4 fluorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 4 chlorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 3 chlorophenyl 1H pyrazol 4 yl boronic acid 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 4 fluorophenyl 1H pyrazol 4 yl boronic acid 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl morpholine 2 piperidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl propan 2 ol

2 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 4 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 carbonitrile 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 isopropoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 ethoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 chloro 2 fluoropyridin 3 yl boronic acid 5 fluoro 2 methoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 ol 3 chloro 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 3 difluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 3 dichloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl picolinonitrile 2 methoxy 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 amine 2 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methylthio 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl pyridine 4 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 ethoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 ethoxycarbonyl 5 fluorophenylboronic acid 4 methoxy 3 trifluoromethyl phenylboronic acid 3 fluoro 5 methylphenylboronic acid 3 fluoro 5 isobutoxyphenylboronic acid 3 fluoro 5 methoxyphenylboronic acid 3 fluoro 5 hydroxyphenylboronic acid 2 cyano 4 fluorophenylboronic acid

4 allyloxy phenylboronic acid 4 2 methoxy 2 oxoethyl phenylboronic acid 3 chloro 5 methoxycarbonyl phenylboronic acid 3 methoxycarbonyl 5 methylphenylboronic acid 4 chloro 3 methoxyphenylboronic acid 4 methyl 3 4 dihydro 2H benzo b 1 4 oxazin 7 ylboronic acid 3 3 bromopropylcarbamoyl phenylboronic acid 2 fluoro 5 methoxycarbonyl phenylboronic acid 3 methyl 4 propoxyphenylboronic acid 3 dipropylcarbamoyl phenylboronic acid 3 propoxycarbonyl phenylboronic acid 5 chloro 2 hydroxyphenylboronic acid 4 hydrazinecarbonyl phenylboronic acid 4 benzoylphenylboronic acid 2 ethoxy 6 fluorophenylboronic acid 3 1H pyrazol 1 yl phenylboronic acid 4 benzyloxy 3 methylphenylboronic acid 3 bromo 5 fluorophenylboronic acid 2 isobutoxyphenylboronic acid 4 2 dimethylamino ethylcarbamoyl phenylboronic acid hydrochloride 2 chloro 5 formylphenylboronic acid 4 borono 2 methoxybenzoic acid 2 3 difluoro 4 pentyloxy phenylboronic acid 8 methylquinolin 5 ylboronic acid 3 ethylcarbamoyl phenylboronic acid 3 butylcarbamoyl phenylboronic acid 3 amino 4 methoxyphenylboronic acid hydrochloride 5 chloro 2 fluoro 4 methoxyphenylboronic acid 4 3 methoxy 3 oxopropyl phenylboronic acid 3 3 methoxy 3 oxopropyl phenylboronic acid

4 3 ethoxy 3 oxoprop 1 enyl phenylboronic acid 4 ethoxy 3 fluorophenylboronic acid 3 benzylcarbamoyl phenylboronic acid 4 isopropylcarbamoyl phenylboronic acid 2 3 5 6 tetrafluorophenylboronic acid 2 methoxy 5 trifluoromethyl phenylboronic acid 4 propionylphenylboronic acid 3 propionylphenylboronic acid 4 pentyloxy phenylboronic acid 3 methylcarbamoyl phenylboronic acid 4 ethylbiphenyl 4 ylboronic acid 6 hydroxynaphthalen 2 ylboronic acid 2 5 difluoro 4 methoxyphenylboronic acid 3 chloro 2 6 difluorophenylboronic acid 4 tert butoxycarbonylamino 3 methoxyphenylboronic acid 4 butylcarbamoyl phenylboronic acid 4 methoxycarbonylamino phenylboronic acid 2 methylquinolin 5 ylboronic acid 3 ethoxy 2 fluorophenylboronic acid 4 chloro 3 methoxycarbonyl phenylboronic acid 5 chloro 2 fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 3 trifluoromethyl pyridine 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 5 trifluoromethyl pyridine 5 chloro 2 fluorophenylboronic acid 3 methoxymethoxy phenylboronic acid 3 chloro 4 methoxyphenylboronic acid 5 methoxy 2 trifluoromethyl phenylboronic acid 2 3 4 trifluorophenylboronic acid 2 4 6 trichlorophenylboronic acid 3 2 methoxy 2 oxoethyl phenylboronic acid