3 acetylphenylboronic acid 8 bromoquinolin 2 1H one 3 4 Dichloro 6 trifluoromethyl toluene 3 Fluoro 4 nitrobenzyl bromide 5 Methoxy 2 methylbenzoic acid 3 Fluoro 4 iodonitrobenzene 2 Bromo 6 fluoroanisole 2 Chloro 2 4 difluoroacetophenone 1 5 Trifluoromethyl pyridin 2 yl piperazine 1 3 5 Triisopropylbenzene 2 Amino 4 chloro 5 formylthiophene 3 carbonitrile 4 Bromo 2 fluorothiophenol 3 Fluoroacetanilide 3 Trifluoromethyl phenylacetic acid 2 3 Dibromoacetophenone 2 Hydroxy 3 methylbenzaldehyde 5 Bromo 2 chlorobenzyl cyanide 2 5 Dimethylbenzyl chloride 2 4 5 Trimethylbenzoic acid 4 Fluoro 2 methylaniline 5 Bromophthalide 1 1 Thiocarbonyldiimidazole 4 Acetylamino 2 2 6 6 tetramethylpiperidin 1 oxyl 3 4 Dichloropyridine 3 5 Dichlorobenzaldehyde 2 Amino 3 methoxybenzoic acid 3 Fluorobenzonitrile 1 Naphthalenesulfonyl fluoride 8 2 Chlorophenyl 2 methyl 6 4 methylpiperazin 1 yl 9 tetrahydro 2H pyran 4 yl 9H purine 3 fluoro 5 methylpyridin 2 amine

4 tert butyl 15 fluoro 3 5 10 triazatetracyclo 11 4 0 0² ⁶ 0⁷ ¹² heptadeca 1 13 2 6 4 7 12 8 14 16 heptaen 11 one 6 bromo 5 fluoro 1 methyl 1H indazole 4 fluoro 1H pyrrolo 2 3 b pyridin 6 ol 2 bromo 4 5 difluoropyridine 4 chloro 5 trifluoromethyl 1H pyrrolo 2 3 b pyridine 7 bromo 2 methoxyquinoxaline 2s 2 fluoromethyl pyrrolidine hydrochloride 4 methoxy 5 6 7 8 tetrahydropyrido 3 4 d pyrimidine hydrochloride 2 4 dichloro 3 nitroquinoline 4 amino 2 3 bithiophene 5 carboxamide 2 hydroxy 3 trifluoromethyl phenylboronic acid 4 4 5 5 tetramethyl 2 3 methylthiophen 2 yl 1 3 2 dioxaborolane 1 nitroisoquinoline 3 bromo 5 fluorophenyl methyl sulfane 1 1 phenylethyl piperidin 4 one 4 fluoro 3 methylphenylboronic acid 6 bromo 3 chloropyrazin 2 amine 5 bromo 1 chloroisoquinoline 2 6 Dichloro 3 nitrotoluene 2 Fluoro 6 nitrobenzyl bromide 3 Fluoro 2 iodonitrobenzene 2 Bromo 3 fluoroanisole 2 Chloro 1 2 5 difluorophenyl ethanone 1 4 Trifluoromethyl benzyl piperazine 4 Cyano 3 fluoroacetophenone 3 5 Bis trifluoromethyl thiophenol 2 amino 5 Bromo 3 methoxypyrazine 2 6 Dimethylacetanilide 4 Hydroxy 3 methoxybenzaldehyde 2 Bromo 4 chlorobenzyl cyanide

3 4 5 Trimethoxybenzoic acid 2 4 Dimethylbenzyl chloride 2 Trifluoromethyl phenylacetic acid 2 Methyl 1 octylindole 4 fluoro 3 nitrotoluene 9 Bromoanthracene 1 Acetoxy 4 fluorobenzene 5 Bromo 2 chlorobenzonitrile 2 Methoxy 5 picoline 4 Bromo 3 trifluoromethyl benzonitrile 2 7 ethoxy 4 3 fluorophenyl 1 oxo 1 2 dihydrophthalazin 2 yl N methyl N 2 methyl 1 3 benzoxazol 6 yl acetamide 3s 4r rel 4 boc amino 3 fluoropiperidine 6 bromo 4 fluoro 1H pyrrolo 2 3 b pyridine 6 bromo 5 fluoro 3 methyl 1H indazole 4 4 trifluoromethyl phenyl phenyl methanamine 2 bromo 5 fluoro 4 iodopyridine 2R pyrrolidine 2 carbonitrile trifluoroacetate 4 Amino 6 chloro 2 methoxypyrimidine 1 3 iodothiophen 2 yl ethanone 2 4 fluorophenyl 3 oxo 2 3 dihydropyridazine 4 carboxylic acid 2 iodonicotinonitrile 4 cyano 3 methoxyphenylboronic acid 1 2 methylbenzo d oxazol 6 yl 3 1 5 naphthyridin 4 yl urea 4 chloro 2 3 dimethylpyridine 4 chloro 7 8 dimethoxyquinazoline 2 bromo N N dimethylpyrimidin 5 amine 3 5 dimethoxyisonicotinic acid 5 chloro 3 methylbenzo b thiophene 3 chloro 4 methoxyphenylboronic acid 5 bromoisoquinolin 1 amine

3 5 Dichlorotoluene 2 Fluoro 5 nitronbenzyl alcohol 5 Bromo 2 3 difluorophenol 2 Fluoro 5 iodonitrobenzene 4 Chloro 2 2 2 trifluoroacetophenone 4 4 Trifluoromethoxy phenoxy piperidine 1 Acetyl 4 piperidinecarboxylic acid 2 Nitro 1 3 5 tri tert butylbenzene 3 Cyanoacetophenone 3 Hydroxy 4 methoxybenzaldehyde 4 Bromobenzyl cyanide 2 6 Difluorobenzyl chloride 2 Trifluoromethyl benzoic acid 4 Trifluoromethoxy phenylacetic acid 1 3 5 Triazine 1 3 5 tributylhexahydro 4 Fluoro 2 nitrotoluene 4 Trifluoromethyl biphenyl 4 carbaldehyde 2 Methoxy 5 nitro 4 picoline 2 Fluoro 6 iodoanisole 2 4 5 Triiodoimidazole 4 Bromo 2 trifluoromethyl benzonitrile 1 4 fluorophenyl methyl cyclopropane 1 carboxylic acid 4 fluoro 2 methyl 1H pyrrolo 2 3 b pyridine 2S pyrrolidine 2 carbonitrile trifluoroacetate 4 fluoro 1H pyrrolo 2 3 b pyridine 6 carbonitrile 5 5 difluorooxan 3 amine 6 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl indolin 2 one 2 3 trifluoromethyl phenoxy nicotinic acid 2 iodonicotinic acid 2 anthracen 9 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane